SCHEMBL4276353

SCHEMBL4276353

Brc1ccc(P(Br)Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.53
ALDH1A1 P00352 4/20 0.40
ALOX15 P16050 2/20 0.40
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 1/20 0.37
CA2 P00918 4/20 0.35
CA1 P00915 3/20 0.35
TSHR P16473 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
HTR2A P28223 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
SLC22A2 O15244 1/20 0.31
SLC22A1 O15245 1/20 0.31
SLC22A3 O75751 1/20 0.31
PLAU P00749 1/20 0.31
MAPT P10636 1/20 0.31
PLCG1 P19174 1/20 0.31
IDO1 P14902 1/20 0.31
GLB1 P16278 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3757571 0.76 CYP2A6 (0.57) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL18508 0.73
SCHEMBL11916255 0.71 CYP2A6 (0.50) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL2884210 0.71 CYP2A6 (0.50) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL11770595 0.71 CYP2A6 (0.50) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL9717534 0.71 CYP2A6 (0.50) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL972975 0.69
SCHEMBL7613201 0.69 CYP2A6 (0.47) CYP2A6ALDH1A1ALOX15MAPK1TDP1
SCHEMBL3138002 0.69
Methane SCHEMBL21489530 0.69 CYP2A6 (0.89) CYP2A6ALDH1A1ALOX15MAPK1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9871213-B2 Organic electroluminescent device MERCK PATENT GMBH (DE) 2018-01-16 US disclosed
US-20160322570-A1 ORGANIC ELECTROLUMINESCENT DEVICE MERCK PATENT GMBH (DE) 2016-11-03 US disclosed
US-9403849-B2 Organic electroluminescent device and boric acid and borinic acid derivatives used therein MERCK PATENT GMBH (DE) 2016-08-02 US disclosed
US-20150322091-A1 ORGANIC ELECTROLUMINESCENT DEVICE AND BORIC ACID AND BORINIC ACID DERIVATIVES USED THEREIN MERCK PATENT GMBH (DE) 2015-11-12 US disclosed
US-8674141-B2 Organic electroluminescent device and boric acid and borinic acid derivatives used therein MERCK PATENT GMBH (DE) 2014-03-18 US disclosed
US-20090134384-A1 ORGANIC ELECTROLUMINESCENT DEVICE AND BORIC ACID AND BORINIC ACID DERIVATIVES USED THEREIN MERCK PATENT GMBH (DE) 2009-05-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090134384-A1 ORGANIC ELECTROLUMINESCENT DEVICE AND BORIC ACID AND BORINIC ACID DERIVATIVES USED THEREIN BTD, ERG, OR10J3 CYP2A6 2674/4885ALDH1A1 857/4885ALOX15 1041/4885
US-20160322570-A1 ORGANIC ELECTROLUMINESCENT DEVICE OR10J3, BTD, ERG CYP2A6 3477/4885ALDH1A1 1034/4885ALOX15 1567/4885
US-20150322091-A1 ORGANIC ELECTROLUMINESCENT DEVICE AND BORIC ACID AND BORINIC ACID DERIVATIVES USED THEREIN BTD, ERG, OR10J3 CYP2A6 2674/4885ALDH1A1 857/4885ALOX15 1041/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.