SCHEMBL4277759

SCHEMBL4277759

Cc1nc(Cc2ccc(Cl)cc2)sc1NC(=O)c1ccc2c(c1)CCNC2

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGER1 P34995 3/20 0.48
SLC2A1 P11166 2/20 0.45
WNT1 P04628 3/20 0.43
GSK3B P49841 3/20 0.43
DYRK1A Q13627 3/20 0.43
CLK2 P49760 2/20 0.43
CLK3 P49761 2/20 0.43
F2 P00734 1/20 0.42
PLG P00747 1/20 0.42
PLAU P00749 1/20 0.42
PLAT P00750 1/20 0.42
KLKB1 P03952 1/20 0.42
PRSS1 P07477 1/20 0.42
MAP3K5 Q99683 1/20 0.42
GPR52 Q9Y2T5 1/20 0.41
CYP3A4 P08684 1/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4279956 0.99 PTGER1 (0.48) PTGER1SLC2A1WNT1GSK3BDYRK1A
SCHEMBL4276192 0.84 HPGD (0.58) PTGER1SLC2A1WNT1GSK3BDYRK1A
Hydrochloric Acid SCHEMBL4287252 0.83 HPGD (0.57) PTGER1SLC2A1WNT1GSK3BDYRK1A
SCHEMBL3737875 0.82 L3MBTL1 (0.59) SLC2A1CYP3A4KDM4EALDH1A1MAPT
SCHEMBL13573319 0.82 SLC2A1 (0.49) SLC2A1F2PLGPLAUPLAT
SCHEMBL4289707 0.82 PTGER1 (0.46) PTGER1SLC2A1WNT1GSK3BDYRK1A
Hydrochloric Acid SCHEMBL3734681 0.81 L3MBTL1 (0.58) PTGER1SLC2A1CYP3A4KDM4EALDH1A1
Hydrochloric Acid SCHEMBL4279816 0.81 PTGER1 (0.46) PTGER1SLC2A1WNT1GSK3BDYRK1A
SCHEMBL4285351 0.79 MAPT (0.46) PTGER1SLC2A1WNT1GSK3BDYRK1A
SCHEMBL13573316 0.78 ESR2 (0.48) PTGER1MAP3K5HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed