SCHEMBL4285351

SCHEMBL4285351

CCc1nc(NC(=O)c2ccc3c(c2)CCNC3)sc1Cc1ccc(Cl)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.46
KDM4E B2RXH2 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
HTT P42858 1/20 0.46
SLC2A1 P11166 2/20 0.43
WNT1 P04628 3/20 0.43
GSK3B P49841 3/20 0.43
DYRK1A Q13627 3/20 0.43
PTGER1 P34995 2/20 0.43
CYP3A4 P08684 1/20 0.41
F2 P00734 1/20 0.41
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
KLKB1 P03952 1/20 0.41
PRSS1 P07477 1/20 0.41
CLK2 P49760 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4287368 0.99 MAPT (0.45) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL4284197 0.94 MAPT (0.45) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL4276192 0.89 HPGD (0.58) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
Hydrochloric Acid SCHEMBL4287252 0.89 HPGD (0.57) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL4289707 0.88 PTGER1 (0.46) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
Hydrochloric Acid SCHEMBL4279816 0.87 PTGER1 (0.46) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL3737875 0.81 L3MBTL1 (0.59) MAPTKDM4ESMN1; SMN2ALDH1A1SLC2A1
SCHEMBL4288907 0.81 HPGD (0.52) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
SCHEMBL4282184 0.80 HPGD (0.52) MAPTKDM4ESMN1; SMN2ALDH1A1LMNA
Hydrochloric Acid SCHEMBL3734681 0.80 L3MBTL1 (0.58) MAPTKDM4ESMN1; SMN2ALDH1A1SLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO claimed
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed