SCHEMBL4279451

SCHEMBL4279451

NC(=O)c1nccc2ccccc12.O=C(O)c1nccc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 2/20 0.50
CNR2 P34972 5/20 0.48
PLAU P00749 3/20 0.46
PLG P00747 1/20 0.46
F12 P00748 1/20 0.46
NCF1 P14598 1/20 0.46
NOS3 P29474 1/20 0.46
NOS1 P29475 1/20 0.46
NOS2 P35228 1/20 0.46
BACE1 P56817 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HDAC9 Q9UKV0 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4282133 0.98 RAB9A (0.49) RAB9ACNR2PLAUPLGF12
SCHEMBL29358323 0.93 CNR2 (0.53) RAB9ACNR2PLAUPLGF12
SCHEMBL111310 0.93 CNR2 (0.53) RAB9ACNR2PLAUPLGF12
Hydrochloric Acid SCHEMBL4433615 0.91 CNR2 (0.51) RAB9ACNR2PLAUPLGF12
Naphthalene SCHEMBL10758679 0.91 CNR2 (0.51) RAB9ACNR2PLAUPLGF12
SCHEMBL28198741 0.91 CNR2 (0.51) RAB9ACNR2PLAUPLGF12
SCHEMBL287165 0.91 RAB9A (0.56) RAB9ACNR2PLAUPLGF12
SCHEMBL22664584 0.90 RAB9A (0.55) RAB9ACNR2PLAUPLGF12
Hydrochloric Acid SCHEMBL3294760 0.90 RAB9A (0.55) RAB9ACNR2PLAUPLGF12
Ammonia Solution, Strong SCHEMBL28091481 0.90 RAB9A (0.55) RAB9ACNR2PLAUPLGF12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150196-A1 N-THIAZOLYL-1, 2, 3, 4-TETRAHYDRO-6-ISOQUINOLINECARBOXAMIDE DERIVATIVES AS INHIBITORS OF STEAROYL COENZYME A DESATURASE SMITHKLINE BEECHAM CORPORATION (US) 2009-12-17 WO disclosed