SCHEMBL4280065

SCHEMBL4280065

Clc1c(-c2ccccc2)[nH]c2cc[c]cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.53
MAOB P27338 2/20 0.53
ESR1 P03372 3/20 0.46
ESR2 Q92731 3/20 0.46
CYP19A1 P11511 1/20 0.41
NPSR1 Q6W5P4 1/20 0.39
DYRK1A Q13627 1/20 0.39
CNR1 P21554 1/20 0.37
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL695828 0.83 MAPK14 (0.40) MAOAMAOBKDM4EMAPTHTR2A
SCHEMBL694066 0.83 ESR1 (0.46) MAOAMAOBESR1ESR2CYP19A1
SCHEMBL695360 0.81 F2 (0.48) MAOAMAOBESR1ESR2CYP19A1
SCHEMBL11339598 0.81 MAOA (0.44) MAOAMAOBESR1ESR2CYP19A1
SCHEMBL31681138 0.81 ESR1 (0.61) MAOAMAOBESR1ESR2CYP19A1
SCHEMBL25035 0.74 ALDH1A1 (0.61) MAOAMAOBALDH1A1KDM4EMEN1
SCHEMBL699697 0.72 ESR1 (0.65) ESR1ESR2ALDH1A1KDM4EMEN1
SCHEMBL11330988 0.71 MAOA (0.44) MAOAMAOBALDH1A1KDM4EMEN1
SCHEMBL4276835 0.71 ESR1 (0.41) MAOAMAOBESR1ESR2CYP19A1
SCHEMBL694496 0.70 ALDH1A1 (0.61) NPSR1DYRK1AALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2120569-A2 SPIROCHROMANON DERIVATIVES Merck & Co., Inc. (US) 2009-11-25 EP disclosed
WO-2008088692-A2 SPIROCHROMANON DERIVATIVES MERCK & CO., INC. (US) 2008-07-24 WO disclosed