SCHEMBL4282209

SCHEMBL4282209

CCCCOC(=O)NC1CCC(O)CC1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.54
MAPK1 P28482 1/20 0.54
HTT P42858 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
EPHX1 P07099 3/20 0.49
EPHX2 P34913 1/20 0.46
NAAA Q02083 2/20 0.44
ACHE P22303 6/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4282204 1.00 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL2575225 1.00 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL4719490 0.93 GAA (0.59) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL13387564 0.93 GAA (0.59) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL30581344 0.90 GAA (0.51) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL16526220 0.88 GAA (0.66) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL8260235 0.87 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL8259162 0.87 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL8257128 0.87 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1
SCHEMBL28019672 0.87 GAA (0.54) GAAMAPK1HTTSMN1; SMN2EPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4665733-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 Bristol-Myers Squibb Company (US) 2025-12-24 EP disclosed
WO-2024173323-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 BRISTOL-MYERS SQUIBB COMPANY (US) 2024-08-22 WO disclosed
EP-4351560-A1 ANTICANCER COMPOUNDS The Regents of the University of California (US) 2024-04-17 EP disclosed
US-11952347-B2 Compounds and methods for the targeted degradation of androgen receptor ARVINAS OPERATIONS, INC. (US) 2024-04-09 US disclosed
WO-2022261204-A1 ANTICANCER COMPOUNDS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-12-15 WO disclosed
US-20220259154-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR ARVINAS OPERATIONS, INC. 2022-08-18 US disclosed
EP-2804851-B1 LACTAM DERIVATES USEFUL AS INHIBITORS OF MUTANT IDH1 AGIOS PHARMACEUTICALS INC (US) 2018-07-18 EP disclosed
EP-2663312-A1 IRAK INHIBITORS AND USES THEREOF Nimbus Iris, Inc. (US) 2013-11-20 EP disclosed
WO-2012097013-A1 IRAK INHIBITORS AND USES THEREOF NIMBUS IRIS, INC. (US) 2012-07-19 WO disclosed
US-7615568-B2 3-[2-(cis-4-aminocyclohexyloxy)-4-methylsulfonylbenzoyl-amino]-N-(5-chloropyridin-2-yl)pyridine-2-carboxamide,; anticoagulant; platelet glycoprotein receptor antagonist; thrombosis; orally; acylation of amino-pyridine by (methylthio)benzoic acid followed by oxidation, alkylation, carbonylation ELI LILLY AND COMPANY (US) 2009-11-10 US disclosed
US-20080108594-A1 Antithrombotic Ethers ELI LILLY AND COMPANY (US) 2008-05-08 US disclosed
EP-1644334-B1 ANTITHROMBOTIC ETHERS LILLY CO ELI (US) 2008-01-02 EP disclosed
EP-1644334-A1 ANTITHROMBOTIC ETHERS Eli Lilly and Company (US) 2006-04-12 EP disclosed
WO-2004108677-A1 ANTITHROMBOTIC ETHERS ELI LILLY AND COMPANY (US) 2004-12-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220259154-A1 COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR AR, ADRM1, CRBN GAA 1082/4885MAPK1 4010/4885HTT 2521/4885
US-11952347-B2 Compounds and methods for the targeted degradation of androgen receptor AR, ADRM1, CRBN GAA 1082/4885MAPK1 4010/4885HTT 2521/4885
US-20080108594-A1 Antithrombotic Ethers F11, SERPINC1, F2 GAA 2082/4885MAPK1 416/4885HTT 4023/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.