SCHEMBL4286325

SCHEMBL4286325

COc1nc(C(F)(F)F)c(C)c(=O)[nH]1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.39
KDM5B Q9UGL1 1/20 0.36
HCAR2 Q8TDS4 4/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KHK P50053 1/20 0.33
PDE3B Q13370 2/20 0.33
PDE3A Q14432 2/20 0.33
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
POLB P06746 2/20 0.31
MEN1 O00255 1/20 0.31
MAPT P10636 1/20 0.31
PABPC1 P11940 1/20 0.31
KMT2A Q03164 1/20 0.31
TNKS O95271 1/20 0.30
TNKS2 Q9H2K2 1/20 0.30
PARP2 Q9UGN5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4284667 0.77 CDK4 (0.43) PDE2AKDM5BKDM4EALDH1A1KHK
SCHEMBL4283741 0.71 L3MBTL1 (0.41) PDE2AKDM5BHCAR2KDM4EALDH1A1
SCHEMBL16787495 0.68 HCAR2 (0.34) HCAR2
SCHEMBL4287126 0.63 KDM5B (0.42) KDM5BMEN1KMT2A
SCHEMBL9582021 0.60 HPGD (0.47) KDM5BALDH1A1
SCHEMBL4282510 0.60 CASR (0.41) KDM5BALDH1A1
SCHEMBL24812797 0.59 MAPT (0.53) HCAR2ALDH1A1PDE3BPDE3AMAPT
SCHEMBL15470617 0.59 ALDH1A1 (0.41) KDM4EALDH1A1POLBMAPTTNKS2
SCHEMBL4369980 0.59 POLB (0.34) KDM4EPOLBMAPT
SCHEMBL5115571 0.59 ALDH1A1 (0.43) HCAR2KDM4EALDH1A1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158258-A1 HERBICIDAL DIHYDRO OXO SIX-MEMBERED AZINYL ISOXAZOLINES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2009-12-30 WO disclosed