Phosmet

Phosmet

SCHEMBL428639

COP(=S)(OC)SCN1C(=O)c2ccccc2C1=O.NC(CCCc1ccccc1)C(=O)O

nearest known ligand 0.63

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.63
MAPT P10636 3/20 0.63
HPGD P15428 2/20 0.63
ALOX15 P16050 2/20 0.63
PLIN1 O60240 1/20 0.63
PLIN5 Q00G26 1/20 0.63
ABHD5 Q8WTS1 1/20 0.63
GRIK1 P39086 1/20 0.46
TSHR P16473 2/20 0.40
MAPK1 P28482 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MMP2 P08253 2/20 0.39
MMP9 P14780 2/20 0.39
CASP3 P42574 1/20 0.38
LTA4H P09960 1/20 0.37
ASAH1 Q13510 1/20 0.36
ELANE P08246 1/20 0.36
NOS1 P29475 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosmet SCHEMBL1663406 0.80 ALDH1A1 (1.00) ALDH1A1MAPTHPGDALOX15PLIN1
Phosmet SCHEMBL29350557 0.80 ALDH1A1 (1.00) ALDH1A1MAPTHPGDALOX15PLIN1
Phosmet SCHEMBL3620 0.80 ALDH1A1 (1.00) ALDH1A1MAPTHPGDALOX15PLIN1
Phosmet SCHEMBL7246728 0.78 ALDH1A1 (0.84) ALDH1A1MAPTHPGDALOX15PLIN1
SCHEMBL2130589 0.73 GRIK1 (0.73) GRIK1MAPK1TDP1LTA4HNOS1
SCHEMBL5082998 0.73 GRIK1 (0.73) GRIK1MAPK1TDP1LTA4HNOS1
SCHEMBL377574 0.73 GRIK1 (0.73) GRIK1MAPK1TDP1LTA4HNOS1
Phosmet SCHEMBL15561615 0.72 ALDH1A1 (0.78) ALDH1A1MAPTHPGDALOX15PLIN1
Hydrochloric Acid SCHEMBL7359673 0.71 GRIK1 (0.71) GRIK1MAPK1TDP1LTA4HNOS1
Hydrochloric Acid SCHEMBL27975738 0.71 GRIK1 (0.71) GRIK1MAPK1TDP1LTA4HNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8883963-B2 Peptidomimetics with glucagon antagonistic and GLP 1 agonistic activities CADILA HEALTHCARE LIMITED (IN) 2014-11-11 US disclosed
US-8383581-B2 Short-chain peptides as parathyroid hormone (PTH) receptor agonist CADILA HEALTHCARE LIMITED (IN) 2013-02-26 US disclosed
US-20120264685-A1 SHORT CHAIN PEPTIDOMIMETICS BASED ORALLY ACTIVE GLP 1 AGONIST AND GLUCAGON RECEPTOR ANTAGONIST CADILA HEALTHCARE LIMITED (IN) 2012-10-18 US disclosed
WO-2012120532-A2 CYCLIC SHORT CHAIN PEPTIDES CADILA HEALTHCARE LIMITED (IN) 2012-09-13 WO disclosed
US-20120108496-A1 SHORT-CHAIN PEPTIDES AS PARATHYROID HORMONE (PTH) RECEPTOR AGONIST CADILA HEALTHCARE LIMITED (IN) 2012-05-03 US disclosed
EP-2231701-B1 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP-1 AGONISTIC ACTIVITIES CADILA HEALTHCARE LTD (IN) 2012-04-18 EP disclosed
EP-2421893-A2 SHORT-CHAIN PEPTIDES AS PARATHYROID HORMONE (PTH) RECEPTOR AGONIST Cadila Healthcare Limited (IN) 2012-02-29 EP disclosed
US-20120021972-A1 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP 1 AGONISTIC ACTIVITIES CADILA HEALTHCARE LIMITED (IN) 2012-01-26 US disclosed
WO-2010128521-A2 SHORT-CHAIN PEPTIDES AS PARATHYROID HORMONE (PTH) RECEPTOR AGONIST CADILA HEALTHCARE LIMITED (IN) 2010-11-11 WO disclosed
EP-2231701-A2 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP-1 AGONISTIC ACTIVITIES Cadila Healthcare Limited (IN) 2010-09-29 EP disclosed
WO-2009125424-A2 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP-1 AGONISTIC ACTIVITIES CADILA HEALTHCARE LIMITED (IN) 2009-10-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108496-A1 SHORT-CHAIN PEPTIDES AS PARATHYROID HORMONE (PTH) RECEPTOR AGONIST PTH1R, GIPR, PTMS ALDH1A1 3467/4885MAPT 4729/4885HPGD 668/4885
US-20120264685-A1 SHORT CHAIN PEPTIDOMIMETICS BASED ORALLY ACTIVE GLP 1 AGONIST AND GLUCAGON RECEPTOR ANTAGONIST GIPR, GLP1R, DPP4 ALDH1A1 2704/4885MAPT 4604/4885HPGD 1540/4885
US-20120021972-A1 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP 1 AGONISTIC ACTIVITIES GLP1R, GPR119, GIPR ALDH1A1 3147/4885MAPT 4741/4885HPGD 2980/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.