SCHEMBL4288131

SCHEMBL4288131

ClOn1ccc2ccccc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 4/20 0.45
CCND1 P24385 4/20 0.45
BIRC5 O15392 1/20 0.42
NOTUM Q6P988 1/20 0.39
HTR6 P50406 2/20 0.39
KMT2A Q03164 2/20 0.37
TSHR P16473 2/20 0.37
RAB9A P51151 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PRKD3 O94806 1/20 0.37
PRKCG P05129 1/20 0.37
PRKCB P05771 1/20 0.37
PRKCA P17252 1/20 0.37
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
PRKCH P24723 1/20 0.37
PRKCI P41743 1/20 0.37
PRKCE Q02156 1/20 0.37
PRKCQ Q04759 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3576716 0.78 CDK4 (0.47) CDK4CCND1NOTUMHTR6KMT2A
SCHEMBL30233726 0.78 CDK4 (0.47) CDK4CCND1NOTUMHTR6KMT2A
SCHEMBL7987460 0.78 CDK4 (0.42) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL22769564 0.77 CDK4 (0.45) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL321199 0.77 CDK4 (0.45) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL29614841 0.77 CDK4 (0.45) CDK4CCND1BIRC5NOTUMHTR6
Hydrochloric Acid SCHEMBL7218572 0.76 CDK4 (0.43) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL10932323 0.74 CDK4 (0.42) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL8995369 0.74 CDK4 (0.42) CDK4CCND1BIRC5NOTUMHTR6
SCHEMBL31276881 0.74 CDK4 (0.39) CDK4CCND1NOTUMKMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090257975-A1 Solid and Semi-Solid Polymeric Ionic Conjugates PFIZER INC 2009-10-15 US disclosed
WO-2006032957-A1 IN VITRO PREDICTIVE METHOD PFIZER PRODUCTS INC. (US) 2006-03-30 WO disclosed
US-20060031021-A1 In vitro predictive method PFIZER INC 2006-02-09 US disclosed
EP-1575616-A2 NOVEL INJECTABLE DEPOT FORMULATIONS Pfizer Products Inc. (US) 2005-09-21 EP disclosed
EP-1562546-A1 DEPOT FORMULATIONS OF ARYLHETEROCYCLIC ACTIVE AGENTS IN THE FORM OF A SUSPENSION Pfizer Products Inc. (US) 2005-08-17 EP disclosed
EP-1556086-A2 SOLID AND SEMI-SOLID POLYMERIC IONIC CONJUGATES Pfizer Products Inc. (US) 2005-07-27 EP disclosed
EP-1556087-A2 LIQUID CONJUGATES OF SOLID PHARMACEUTICALS Pfizer Products Inc. (US) 2005-07-27 EP disclosed
US-20040146562-A1 Depot formulations in the form of a suspension PFIZER INC 2004-07-29 US disclosed
US-20040147532-A1 Liquid conjugates of solid pharmaceuticals PFIZER INC 2004-07-29 US disclosed
US-20040142039-A1 Solid and semi-solid polymeric ionic conjugates PFIZER INC 2004-07-22 US disclosed
US-20040138237-A1 Novel injectable depot formulations PFIZER INC 2004-07-15 US disclosed
WO-2004039411-A2 SOLID AND SEMI-SOLID POLYMERIC IONIC CONJUGATES PFIZER PRODUCTS INC. (GB) 2004-05-13 WO disclosed
WO-2004039410-A2 LIQUID CONJUGATES OF SOLID PHARMACEUTICALS PFIZER PRODUCTS INC. (US) 2004-05-13 WO disclosed
WO-2004037289-A2 NOVEL INJECTABLE DEPOT FORMULATIONS PFIZER PRODUCTS INC. (US) 2004-05-06 WO disclosed
WO-2004037224-A1 DEPOT FORMULATIONS OF ARYLHETEROCYCLIC ACTIVE AGENTS IN THE FORM OF A SUSPENSION PFIZER PRODUCTS INC. (US) 2004-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040138237-A1 Novel injectable depot formulations NPY4R, GLP1R, GPR119 CDK4 317/4885CCND1 2438/4885BIRC5 3459/4885
US-20040146562-A1 Depot formulations in the form of a suspension LPXN, HAMP, GLP1R CDK4 551/4885CCND1 1815/4885BIRC5 3650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.