SCHEMBL4289486

SCHEMBL4289486

CNC(=O)C1Cc2ccccc2C1C(N)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.38
HDAC7 Q8WUI4 2/20 0.38
HDAC5 Q9UQL6 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
ALDH1A1 P00352 2/20 0.36
GAA P10253 2/20 0.36
P2RX7 Q99572 1/20 0.35
HSP90AA1 P07900 1/20 0.34
HSP90AB1 P08238 1/20 0.34
MTNR1A P48039 3/20 0.34
MTNR1B P49286 3/20 0.34
CYP3A4 P08684 3/20 0.34
TSHR P16473 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4286038 0.84 ALDH1A1 (0.41) HDAC4HDAC7HDAC5ALDH1A1GAA
SCHEMBL4283036 0.84 ALDH1A1 (0.41) HDAC4HDAC7HDAC5ALDH1A1GAA
SCHEMBL4289491 0.81 HDAC4 (0.40) HDAC4HDAC7HDAC5HDAC3HDAC1
SCHEMBL14143070 0.76 ALDH1A1 (0.41) ALDH1A1GAA
SCHEMBL562899 0.74 KDM1A (0.42) ALDH1A1GAASIGMAR1
SCHEMBL177215 0.74 ALDH1A1 (0.41) ALDH1A1GAAP2RX7MEN1KMT2A
SCHEMBL2699779 0.74 ALDH1A1 (0.41) ALDH1A1GAAP2RX7MEN1KMT2A
SCHEMBL3092977 0.74 ALDH1A1 (0.41) ALDH1A1GAAP2RX7MEN1KMT2A
SCHEMBL21016972 0.74 P2RX7 (0.52) HDAC4HDAC7HDAC5HDAC3HDAC1
SCHEMBL177088 0.74 ALDH1A1 (0.41) ALDH1A1GAAP2RX7MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009152824-A1 HETEROCYCLIC DERIVATIVES AS IAP BINDING COMPOUNDS NUEVOLUTION A/S (DK) 2009-12-23 WO disclosed