SCHEMBL4290048

SCHEMBL4290048

Cn1cncc1C(N)(c1ccc2[nH]c(=O)cc(Cc3cccc(Cl)c3)c2c1)c1ccc(Cl)s1

nearest known ligand 0.58

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FNTA P49354 14/20 0.58
FNTB P49356 14/20 0.58
PGGT1B P53609 4/20 0.41
CYP3A4 P08684 3/20 0.41
CNR1 P21554 1/20 0.41
RORC P51449 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28782663 0.89 FNTA (0.72) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL2844704 0.89 FNTA (0.72) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4281997 0.86 FNTA (0.60) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4285788 0.86 FNTA (0.60) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4284855 0.81 FNTA (0.48) FNTAFNTBPGGT1BCNR1RORC
SCHEMBL1682751 0.80 FNTA (0.61) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4278951 0.79 FNTA (0.55) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4276938 0.77 FNTA (0.61) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL4282437 0.77 FNTA (0.51) FNTAFNTBPGGT1BCYP3A4CNR1
SCHEMBL6169281 0.76 FNTA (0.79) FNTAFNTBPGGT1BRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020019530-A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents YANG BINGWEI V (US) 2002-02-14 US claimed
WO-2009151683-A2 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS LINK MEDICINE CORPORATION (US) 2009-12-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019530-A1 Heteroaryl-substituted quinolin-2-one derivatives useful as anticancer agents NRAS, CCNA1, KRAS FNTA 855/4885FNTB 2166/4885PGGT1B 692/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.