SCHEMBL4282437

SCHEMBL4282437

CCOc1cccc(Cc2cc(=O)[nH]c3ccc(C(N)(c4ccc(Cl)nc4)c4cncn4C)cc23)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
FNTA P49354 11/20 0.51
FNTB P49356 11/20 0.51
RORC P51449 3/20 0.41
CYP3A4 P08684 3/20 0.39
PGGT1B P53609 4/20 0.36
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1682751 0.92 FNTA (0.61) FNTAFNTBRORCCYP3A4PGGT1B
SCHEMBL4284860 0.90 RORC (0.53) FNTAFNTBRORC
SCHEMBL4278951 0.86 FNTA (0.55) FNTAFNTBRORCCYP3A4PGGT1B
SCHEMBL4285788 0.83 FNTA (0.60) FNTAFNTBCYP3A4PGGT1BCNR1
SCHEMBL4284855 0.83 FNTA (0.48) FNTAFNTBRORCPGGT1BCNR1
SCHEMBL28782663 0.82 FNTA (0.72) FNTAFNTBCYP3A4PGGT1BCNR1
SCHEMBL2844704 0.82 FNTA (0.72) FNTAFNTBCYP3A4PGGT1BCNR1
SCHEMBL4281997 0.79 FNTA (0.60) FNTAFNTBRORCCYP3A4PGGT1B
SCHEMBL6174101 0.77 FNTA (0.67) FNTAFNTBRORCPGGT1B
SCHEMBL3501050 0.77 FNTA (0.84) FNTAFNTBCYP3A4PGGT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009151683-A2 QUINOLINONE FARNESYL TRANSFERASE INHIBITORS FOR THE TREATMENT OF SYNUCLEINOPATHIES AND OTHER INDICATIONS LINK MEDICINE CORPORATION (US) 2009-12-17 WO disclosed