SCHEMBL429041

SCHEMBL429041

Cc1c(F)cncc1-c1nc2ccccc2n1C

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.51
KMT2A Q03164 3/20 0.51
CYP11B2 P19099 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP11B1 P15538 1/20 0.47
KDM4E B2RXH2 9/20 0.47
ALDH1A1 P00352 7/20 0.47
NPC1 O15118 6/20 0.47
RAB9A P51151 6/20 0.47
TP53 P04637 5/20 0.47
GAA P10253 5/20 0.47
PKM P14618 4/20 0.47
HSD17B10 Q99714 3/20 0.47
ALOX15 P16050 1/20 0.47
SMN1; SMN2 Q16637 6/20 0.46
HPGD P15428 4/20 0.46
MAPT P10636 4/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31339766 0.82 MEN1 (0.59) MEN1KMT2ACYP11B2CYP3A4CYP11B1
SCHEMBL17896690 0.81 CYP11B2 (0.46) MEN1KMT2ACYP11B2CYP3A4CYP11B1
SCHEMBL21022943 0.80 MEN1 (0.52) MEN1KMT2ACYP3A4KDM4EALDH1A1
SCHEMBL3714642 0.80 PDE10A (0.56) MEN1KMT2ACYP3A4KDM4EALDH1A1
SCHEMBL17896708 0.75 CYP11B2 (0.68) CYP11B2CYP3A4CYP11B1
SCHEMBL1171430 0.75 MEN1 (0.69) MEN1KMT2ACYP3A4KDM4EALDH1A1
SCHEMBL6298381 0.75 SMN1; SMN2 (0.49) MEN1KMT2ACYP11B2CYP3A4CYP11B1
SCHEMBL27611222 0.73 SMN1; SMN2 (0.48) MEN1KMT2ACYP11B2CYP3A4CYP11B1
SCHEMBL1533895 0.73 KDM4E (0.48) MEN1KMT2ACYP3A4KDM4EALDH1A1
SCHEMBL22344209 0.73 MEN1 (0.54) MEN1KMT2ACYP3A4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2595482-A1 ALDOSTERONE SYNTHASE INHIBITORS Merck Sharp & Dohme Corp. (US) 2013-05-29 EP claimed
WO-2012012478-A1 ALDOSTERONE SYNTHASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2012-01-26 WO claimed