SCHEMBL17896708

SCHEMBL17896708

Cc1c(F)cncc1-c1nc2ccc(F)c(F)c2n1C

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 10/20 0.68
CYP11B1 P15538 8/20 0.46
CYP3A4 P08684 2/20 0.46
CYP19A1 P11511 1/20 0.35
ABL1 P00519 7/20 0.34
KIT P10721 1/20 0.32
PDGFRA P16234 1/20 0.32
SSTR5 P35346 1/20 0.31
LRRK2 Q5S007 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10175463 0.90 CYP11B2 (0.67) CYP11B2CYP11B1CYP3A4SSTR5
SCHEMBL17897047 0.85 CYP11B2 (0.61) CYP11B2CYP11B1CYP3A4
SCHEMBL10175441 0.83 CYP11B2 (0.62) CYP11B2CYP11B1CYP3A4CYP19A1
SCHEMBL463351 0.82 CYP11B2 (0.67) CYP11B2CYP11B1
SCHEMBL10175445 0.81 CYP11B2 (1.00) CYP11B2CYP11B1CYP3A4
SCHEMBL10175451 0.79 CYP11B2 (0.63) CYP11B2CYP11B1
SCHEMBL17896706 0.78 CYP11B2 (0.61) CYP11B2CYP11B1
SCHEMBL460559 0.77 CYP11B2 (0.46) CYP11B2CYP11B1CYP3A4CYP19A1ABL1
SCHEMBL10175449 0.77 CYP11B2 (0.60) CYP11B2CYP11B1
SCHEMBL17896690 0.77 CYP11B2 (0.46) CYP11B2CYP11B1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed
US-9382226-B2 Aldosterone synthase inhibitors MERCK SHARP & DOHME CORP. (US) 2016-07-05 US disclosed