SCHEMBL4292891

SCHEMBL4292891

CCNC(=O)C(=O)N(C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
KMT2A Q03164 1/20 0.36
MCL1 Q07820 1/20 0.34
CHRNB2 P17787 2/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA4 P43681 2/20 0.34
CHRNA3 P32297 1/20 0.34
ALDH1A1 P00352 4/20 0.33
GAA P10253 1/20 0.33
FAAH O00519 1/20 0.33
CYP3A4 P08684 1/20 0.33
PLAAT3 P53816 1/20 0.32
PLAAT5 Q96KN8 1/20 0.32
PLAAT2 Q9NWW9 1/20 0.32
PLAAT4 Q9UL19 1/20 0.32
TSHR P16473 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4297064 0.80 NPC1 (0.44) MMP1MMP2MMP3MMP9MCL1
SCHEMBL1900809 0.79 MMP1 (0.37) MMP1MMP2MMP3MMP9MMP8
SCHEMBL3060269 0.76 MMP1 (0.48) MMP1MMP2MMP3MMP9MMP8
SCHEMBL2791486 0.75 MMP1 (0.34) MMP1MMP2MMP3MMP9MMP8
SCHEMBL27871351 0.75 MMP1 (0.34) MMP1MMP2MMP3MMP9MMP8
SCHEMBL7776613 0.73 FAAH (0.34) MMP1MMP2MMP3MMP9MMP8
SCHEMBL9298297 0.73 MMP1 (0.33) MMP1MMP2MMP3MMP9MMP8
SCHEMBL4301028 0.73 CYP2D6 (0.50) MMP1MMP8KMT2ACHRNB2CHRNB4
SCHEMBL967318 0.72
SCHEMBL8172250 0.72

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100341949-C 1, 1-dimethyl-3-propanesulfonic indole-1 '- (N, N-dimethyl amino ethylamino) -3' -ethyl-imidazolyl-carbocyanine dye and preparation method and application thereof RIKAGAKU KENKYUSHO (CN) 2007-10-10 CN claimed
CN-1752149-A 1, 1-dimethyl-3-propanesulfonic indole-1 '- (N, N-dimethyl amino ethylamino) -3' -ethyl-imidazolyl-carbocyanine dye and preparation method and application thereof RIKAGAKU KENKYUSHO (CN) 2006-03-29 CN claimed
WO-2022056447-A1 CARBOXYLIC ACID-CONTAINING COMPOUNDS AS MODULATORS OF BIS-PHOSPHOGLYCERATE MUTASE FOR THE TREATMENT OF SICKLE CELL DISEASE GENZYME CORPORATION (US) 2022-03-17 WO disclosed
WO-2010042391-A2 HIV INTEGRASE INHIBITORS MERCK SHARP & DOHME CORP. (US) 2010-04-15 WO disclosed
WO-2010042392-A2 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2010-04-15 WO disclosed
US-20090221571-A1 HIV INTEGRASE INHIBITORS MSD ITALIA S.R.L. (IT) 2009-09-03 US disclosed
CN-100341949-C 1, 1-dimethyl-3-propanesulfonic indole-1 '- (N, N-dimethyl amino ethylamino) -3' -ethyl-imidazolyl-carbocyanine dye and preparation method and application thereof RIKAGAKU KENKYUSHO (CN) 2007-10-10 CN disclosed
CN-1752149-A 1, 1-dimethyl-3-propanesulfonic indole-1 '- (N, N-dimethyl amino ethylamino) -3' -ethyl-imidazolyl-carbocyanine dye and preparation method and application thereof RIKAGAKU KENKYUSHO (CN) 2006-03-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090221571-A1 HIV INTEGRASE INHIBITORS TYMP, CDK2, TYMS MMP1 2480/4885MMP2 2733/4885MMP3 3446/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.