SCHEMBL4302952

SCHEMBL4302952

CC(C)(C)OC(=O)N1CCC(Oc2cc3c(=O)[nH]c(-c4cccc(Cl)c4)cn3c2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1B P47901 4/20 0.46
STS P08842 1/20 0.43
CACNB4 O00305 2/20 0.43
CACNA1A O00555 2/20 0.43
CACNA1G O43497 2/20 0.43
CACNG3 O60359 2/20 0.43
CACNA1F O60840 2/20 0.43
CACNA1H O95180 2/20 0.43
CACNB3 P54284 2/20 0.43
CACNA2D1 P54289 2/20 0.43
CACNG7 P62955 2/20 0.43
CACNA1B Q00975 2/20 0.43
CACNA1D Q01668 2/20 0.43
CACNB1 Q02641 2/20 0.43
CACNG1 Q06432 2/20 0.43
CACNB2 Q08289 2/20 0.43
CACNA1S Q13698 2/20 0.43
CACNA1C Q13936 2/20 0.43
CACNA1E Q15878 2/20 0.43
CACNA2D4 Q7Z3S7 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4311903 0.88 AVPR1B (0.48) AVPR1BSTSCHEK2GPR119TNKS
SCHEMBL4310057 0.88 AVPR1B (0.49) AVPR1BSTSCHEK2GPR119TP53
SCHEMBL4303339 0.77 AVPR1B (0.79) AVPR1B
SCHEMBL3171016 0.77 STS (0.57) STSCACNB4CACNA1ACACNA1GCACNG3
SCHEMBL29731062 0.77 STS (0.57) STSCACNB4CACNA1ACACNA1GCACNG3
SCHEMBL3962648 0.77 STS (0.48) STSGPR119TP53POLB
SCHEMBL4310061 0.77 AVPR1B (0.54) AVPR1B
SCHEMBL4311907 0.76 AVPR1B (0.52) AVPR1B
SCHEMBL8018250 0.74 TNKS (0.46) TNKSPARP1TNKS2
SCHEMBL2793124 0.71 GPR119 (0.65) STSCACNB4CACNA1ACACNA1GCACNG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed