SCHEMBL4303399

SCHEMBL4303399

COC(=O)c1cc(OCCCO[Si](C)(C)C(C)(C)C)cn1CC(=O)c1ccc(F)c(Cl)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.37
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
CASP3 P42574 1/20 0.36
KMT2A Q03164 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
HTR1A P08908 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 1/20 0.35
F2 P00734 1/20 0.34
PLAU P00749 1/20 0.34
KLKB1 P03952 1/20 0.34
ELANE P08246 1/20 0.34
THRB P10828 1/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4304235 0.88 MAPT (0.37) LMNAMAPTKMT2AALDH1A1KDM4E
SCHEMBL4301399 0.88 CYP1A2 (0.34) LMNAALDH1A1KDM4E
SCHEMBL4311072 0.86 MRGPRX4 (0.37) LMNAMEN1KMT2AALDH1A1
SCHEMBL4302813 0.84 ALDH1A1 (0.35) MAPTMEN1KMT2AALDH1A1KDM4E
SCHEMBL4304477 0.83 TP53BP1 (0.38) MAPTKMT2AALDH1A1KDM4E
SCHEMBL4302849 0.82 MCL1 (0.35) LMNAALDH1A1KDM4E
SCHEMBL4305020 0.77 LMNA (0.46) LMNAMAPTMEN1CASP3KMT2A
SCHEMBL4302638 0.76 RXFP1 (0.37) LMNAMAPTMEN1KMT2AHTR1A
SCHEMBL4311981 0.75 LMNA (0.44) LMNAMAPTMEN1CASP3KMT2A
SCHEMBL13125216 0.72 MAPT (0.44) MAPTMEN1KMT2AKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009130231-A1 PYRROLO [1, 2-A] PYRAZINE DERIVATIVES AS VASOPRESSIN VIB RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-10-29 WO disclosed