SCHEMBL4317671

SCHEMBL4317671

Cc1cncc(NC(=O)c2cccc(CCNc3cncc(Cl)n3)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 11/20 0.53
RET P07949 1/20 0.53
PDGFRB P09619 1/20 0.53
KIT P10721 1/20 0.53
SRC P12931 1/20 0.53
PDGFRA P16234 1/20 0.53
FLT1 P17948 1/20 0.53
FLT4 P35916 1/20 0.53
KDR P35968 1/20 0.53
FRK P42685 1/20 0.53
DDR1 Q08345 1/20 0.53
BRAF P15056 2/20 0.44
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43
MAPT P10636 1/20 0.42
GSK3B P49841 1/20 0.42
CYP2C9 P11712 1/20 0.41
KCNQ3 O43525 2/20 0.41
KCNQ2 O43526 2/20 0.41
HRH1 P35367 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324513 0.88 CSF1R (0.66) CSF1RRETPDGFRBKITSRC
SCHEMBL4323640 0.88 CSF1R (0.66) CSF1RRETPDGFRBKITSRC
SCHEMBL4323633 0.81 CYP4F2 (0.53) CSF1RRETPDGFRBKITSRC
SCHEMBL4314900 0.81 CSNK2A2 (0.48) CSF1RBRAF
SCHEMBL27167178 0.81 CSF1R (0.67) CSF1RRETPDGFRBKITSRC
SCHEMBL4318196 0.80 CSF1R (0.66) CSF1RRETPDGFRBKITSRC
SCHEMBL13340052 0.79 CSF1R (0.79) CSF1RRETPDGFRBKITSRC
SCHEMBL3474648 0.79 CSF1R (0.79) CSF1RRETPDGFRBKITSRC
SCHEMBL13340335 0.78 CSF1R (0.65) CSF1RRETPDGFRBKITSRC
SCHEMBL13340328 0.78 CSF1R (0.65) CSF1RRETPDGFRBKITSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099774-A1 INHIBITORS OF KINASE ACTIVITY Cytopia Research Pty Ltd (AU) 2009-09-16 EP disclosed
WO-2008058341-A1 INHIBITORS OF KINASE ACTIVITY CYTOPIA RESEARCH PTY LTD (AU) 2008-05-22 WO disclosed