SCHEMBL4327907

SCHEMBL4327907

CC(C)c1ccc(CNC=O)cn1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 2/20 0.43
ADH1C P00326 2/20 0.43
ADH1A P07327 2/20 0.43
ADH7 P40394 1/20 0.43
PANK3 Q9H999 2/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
PRMT5 O14744 2/20 0.32
WDR77 Q9BQA1 2/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
SLC22A12 Q96S37 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNA1H O95180 1/20 0.31
CNR2 P34972 1/20 0.31
KCNH2 Q12809 1/20 0.31
CACNA1I Q9P0X4 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12986309 0.79 ESR1 (0.39) PANK3ESR1ESR2NPC1RAB9A
SCHEMBL20994112 0.79 ESR1 (0.39) PANK3ESR1ESR2NPC1RAB9A
SCHEMBL4334859 0.76 ACACB (0.53) ACACBACACA
SCHEMBL19323038 0.75 KMT2A (0.47) PANK3NPC1RAB9AKMT2A
SCHEMBL21267702 0.75 KMT2A (0.45) NPC1RAB9AKMT2ACNR2CHRNA7
SCHEMBL19650817 0.75 MEN1 (0.42) RAB9AMEN1KMT2A
SCHEMBL21414391 0.75 L3MBTL1 (0.36) PANK3ESR1ESR2NPC1RAB9A
SCHEMBL22876954 0.75 ALDH1A1 (0.34) PANK3ESR1ESR2NPC1RAB9A
SCHEMBL21266984 0.74 CA1 (0.47) CHRNA7
SCHEMBL7783116 0.74 KDM4E (0.54) ADH1BADH1CADH1AADH7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145720-A1 ISOINDOLINE DERIVATIVES COMPRISING ADDITIONAL HETEROCYCLIC GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed
WO-2009145720-A1 ISOINDOLINE DERIVATIVES COMPRISING ADDITIONAL HETEROCYCLIC GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO disclosed