SCHEMBL4331746

SCHEMBL4331746

Cc1ccc(CCNC(=O)C2c3ccccc3C(=O)N2C2CCC(F)(F)CC2)s1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.56
SCN5A Q14524 5/20 0.56
KCNH2 Q12809 4/20 0.56
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
FPR1 P21462 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
METAP2 P50579 1/20 0.42
ALDH1A1 P00352 1/20 0.41
MAPT P10636 2/20 0.40
KMT2A Q03164 2/20 0.38
KCNA5 P22460 1/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13579102 0.80 SCN9A (0.51) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL13577808 0.75 SCN9A (0.80) SCN9ASCN5AKCNH2SMN1; SMN2FPR1
SCHEMBL4317569 0.74 SCN9A (0.56) SCN9ASCN5AKCNH2TSHRALDH1A1
SCHEMBL4318494 0.74 SCN9A (0.57) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL4321569 0.73 SCN9A (0.79) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL4331776 0.72 SCN9A (0.65) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL3745317 0.72 FPR1 (0.67) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL4325285 0.71 SCN9A (1.00) SCN9ASCN5AKCNH2KCNA5
SCHEMBL3750893 0.70 TSHR (0.61) SCN9ASCN5AKCNH2TSHRSMN1; SMN2
SCHEMBL3745336 0.70 TSHR (0.61) SCN9ASCN5AKCNH2TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009145720-A1 ISOINDOLINE DERIVATIVES COMPRISING ADDITIONAL HETEROCYCLIC GROUPS AND THEIR USE IN THE TREATMENT OF PAIN DISORDERS ASTRAZENECA AB (SE) 2009-12-03 WO claimed