SCHEMBL4336440

SCHEMBL4336440

CC(C)COC(=O)N[C@@H](Cc1cccc(F)c1)CN1C(=O)c2ccccc2C1=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
RAB9A P51151 2/20 0.41
CYP3A4 P08684 1/20 0.41
PIN1 Q13526 3/20 0.40
HTT P42858 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 2/20 0.39
MEN1 O00255 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
UBE2N P61088 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
PLA2G1B P04054 1/20 0.39
ATG4B Q9Y4P1 1/20 0.39
KDM4E B2RXH2 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL683030 0.85 CTSS (0.52) HTTALDH1A1LMNATSHRUBE2N
SCHEMBL4379672 0.85 KMT2A (0.43) CYP2D6CYP2C9CYP2C19RAB9ACYP3A4
SCHEMBL12544607 0.84 CA12 (0.39) CYP2D6CYP2C9CYP2C19RAB9APIN1
SCHEMBL2636369 0.83 PIN1 (0.43) PIN1L3MBTL1ALDH1A1MEN1GAA
SCHEMBL4374776 0.82 CYP3A4 (0.48) CYP2D6CYP2C9CYP2C19RAB9ACYP3A4
SCHEMBL4322435 0.82 PIN1 (0.51) CYP2D6CYP2C9CYP2C19RAB9ACYP3A4
SCHEMBL4583413 0.82 KMT2A (0.50) CYP2D6CYP2C9CYP2C19RAB9ACYP3A4
SCHEMBL4381682 0.78 KMT2A (0.43) CYP2D6CYP2C9CYP2C19RAB9ACYP3A4
SCHEMBL14870407 0.76 ATM (0.47) HTTALDH1A1HPGDMAPK1
SCHEMBL14870379 0.75 TDP1 (0.47) L3MBTL1ALDH1A1MEN1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009158376-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2009-12-30 WO disclosed
WO-2009158374-A2 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2009-12-30 WO disclosed
WO-2009158371-A1 INHIBITORS OF AKT ACTIVITY SMITHKLIKE BEECHAM CORPORATION (US) 2009-12-30 WO disclosed
WO-2009158373-A1 INHIBITORS OF AKT ACTIVITY SMITHKLINE BEECHAM CORPORATION (US) 2009-12-30 WO disclosed