SCHEMBL4339674

SCHEMBL4339674

COc1ccc(C(O)(c2ccc(OC)cc2)[C@H](NC(=O)C(C)(C)C(=O)N[C@H](c2ccccc2)C(O)(c2ccc(OC)cc2)c2ccc(OC)cc2)c2ccccc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.46
ALDH1A1 P00352 3/20 0.45
CYP3A4 P08684 1/20 0.45
GAA P10253 1/20 0.44
KIF11 P52732 3/20 0.43
KMT2A Q03164 3/20 0.42
TP53 P04637 1/20 0.42
CNR2 P34972 1/20 0.42
MEN1 O00255 2/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
GPR88 Q9GZN0 1/20 0.41
ACP3 P15309 1/20 0.41
ATM Q13315 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4344856 0.88 ALDH1A1 (0.48) ALDH1A1CYP3A4GAAKMT2ATP53
SCHEMBL4337659 0.87 CNR1 (0.43) ALDH1A1KMT2ACNR2MEN1HTT
SCHEMBL4340505 0.87 NPC1 (0.46) NPSR1ALDH1A1CYP3A4GAAKMT2A
SCHEMBL4346035 0.85 CNR2 (0.49) NPSR1ALDH1A1CYP3A4GAAKIF11
SCHEMBL4338623 0.85 LMNA (0.48) ALDH1A1GAAKIF11KMT2ATP53
SCHEMBL1154050 0.81 ALDH1A1 (0.43) ALDH1A1CYP3A4GAAKMT2ATP53
SCHEMBL4335644 0.81 KMT2A (0.47) ALDH1A1GAAKMT2AMEN1
SCHEMBL1153400 0.79 ALDH1A1 (0.41) ALDH1A1CYP3A4GAAKMT2ATP53
SCHEMBL1153060 0.79 ALDH1A1 (0.41) ALDH1A1CYP3A4GAAKMT2ATP53
SCHEMBL4340523 0.79 NPSR1 (0.48) NPSR1ALDH1A1CYP3A4GAAKIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7612236-B2 Method for producing optically active bisamidoalcohol compound SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2009-11-03 US disclosed
US-20070100163-A1 Reacting an optically active aminoalcohol compound with a diester compound in the presence of a lithium compound wherein the lithium compound is selected from lithium hydroxide, a lithium alkoxide and a lithium halide; product can be efficiently and inexpensively produced SUMITOMO CHEMICAL COMPANY, LIMITED 2007-05-03 US disclosed
EP-1698616-A1 METHOD FOR PRODUCING OPTICALLY ACTIVE BISAMIDO ALCOHOL COMPOUND Sumitomo Chemical Company, Limited (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070100163-A1 Reacting an optically active aminoalcohol compound with a diester compound in the presence of a lithium compound wherein the lithium compound is selected from lithium hydroxide, a lithium alkoxide and a lithium halide; product can be efficiently and inexpensively produced CCNL2, ARL1, ACSL3 NPSR1 2065/4885ALDH1A1 1303/4885CYP3A4 871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.