SCHEMBL4345928

SCHEMBL4345928

COc1ccc(/C=N/O)cc1OC

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.65
NPC1 O15118 5/20 0.61
RAB9A P51151 5/20 0.61
SMN1; SMN2 Q16637 5/20 0.61
MEN1 O00255 4/20 0.61
KMT2A Q03164 4/20 0.61
NFKB1 P19838 3/20 0.61
NFKB2 Q00653 3/20 0.61
RELA Q04206 3/20 0.61
GFER P55789 1/20 0.60
TP53 P04637 1/20 0.57
POLB P06746 1/20 0.57
PAX8 Q06710 1/20 0.57
KLF5 Q13887 1/20 0.57
HIF1A Q16665 1/20 0.57
TSHR P16473 1/20 0.57
MAPT P10636 4/20 0.56
CYP1A1 P04798 2/20 0.55
CYP1A2 P05177 2/20 0.55
PTGS1 P23219 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2165438 1.00 ALDH1A1 (0.65) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL2165442 1.00 ALDH1A1 (0.65) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4940997 0.86 GAA (0.64) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4941002 0.86 GAA (0.64) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL28969963 0.86 NPC1 (0.64) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL2448826 0.85 ALDH1A1 (0.54) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL4692392 0.85 ALDH1A1 (0.54) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL16221476 0.85 ALDH1A1 (0.54) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL5075035 0.85 ALDH1A1 (0.62) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1
SCHEMBL7990948 0.85 ALDH1A1 (0.62) ALDH1A1NPC1RAB9ASMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111302970-B Preparation method of 3, 4-dimethoxy benzonitrile 河南农业大学 2021-04-27 CN disclosed
CN-111302970-A Preparation method of 3, 4-dimethoxy benzonitrile 河南农业大学 2020-06-19 CN disclosed
US-10174033-B2 N6-substituted adenosine derivatives and N6-substituted adenine derivatives and uses thereof INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2019-01-08 US disclosed
US-20130045942-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES AND N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2013-02-21 US disclosed
EP-2511283-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES, N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF INSTITUTE OF MATERIA MEDICA, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2012-10-17 EP disclosed
US-20110021473-A1 INHIBITORS OF PHOSPHODIESTERASE TYPE-IV RANBAXY LABORATORIES LIMITED 2011-01-27 US disclosed
US-7612069-B2 Acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2009-11-03 US disclosed
US-7273882-B2 Aminoacetamide acyl guanidines as β-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-09-25 US disclosed
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2007-01-18 US disclosed
WO-2007002214-A2 ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
WO-2007002220-A2 AMINOACETAMIDE ACYL GUANIDINES AS BETA-SECRETASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-01-04 WO disclosed
US-20060287287-A1 Aminoacetamide acyl guanidines as beta-secretase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2006-12-21 US disclosed
US-6673800-B2 PREPARATION METHOD THROUGH REDUCTIVE AMINATION REACTION IN THE PRESENCE OF REDUCING AGENT. KOREA INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2004-01-06 US disclosed
US-20020107253-A1 Novel 4,5,-dihydroisoxazolylalkylpiperazine derivatives having selective biological activity at dopamine D3 or D4 receptor, and preparation thereof KOREA ADVANCED INSTITUTE OF SCIENCE AND TECHNOLOGY (KR) 2002-08-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020107253-A1 Novel 4,5,-dihydroisoxazolylalkylpiperazine derivatives having selective biological activity at dopamine D3 or D4 receptor, and preparation thereof DRD4, DRD3, DRD2 ALDH1A1 429/4885NPC1 4430/4885RAB9A 1625/4885
US-20060287287-A1 Aminoacetamide acyl guanidines as beta-secretase inhibitors APP, BACE1, BACE2 ALDH1A1 2529/4885NPC1 1374/4885RAB9A 1220/4885
US-20110021473-A1 INHIBITORS OF PHOSPHODIESTERASE TYPE-IV PDE4A, PDE4B, PDE4C ALDH1A1 306/4885NPC1 4088/4885RAB9A 322/4885
US-20070015754-A1 Acyl guanidines as beta-secretase inhibitors BACE1, APP, BACE2 ALDH1A1 2144/4885NPC1 531/4885RAB9A 558/4885
US-10174033-B2 N6-substituted adenosine derivatives and N6-substituted adenine derivatives and uses thereof ADORA2A, ADORA3, ADORA1 ALDH1A1 1674/4885NPC1 695/4885RAB9A 846/4885
US-20130045942-A1 N6-SUBSTITUTED ADENOSINE DERIVATIVES AND N6-SUBSTITUTED ADENINE DERIVATIVES AND USES THEREOF ADORA2A, ADORA3, ADORA1 ALDH1A1 1674/4885NPC1 695/4885RAB9A 846/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.