SCHEMBL434608

SCHEMBL434608

Clc1ccc(C2CCCCC2)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
TSHR P16473 1/20 0.56
AGTR1 P30556 1/20 0.56
PTGDR2 Q9Y5Y4 8/20 0.46
PTGDR Q13258 5/20 0.46
PTGER2 P43116 1/20 0.46
CEL P19835 2/20 0.46
SIGMAR1 Q99720 2/20 0.43
TMEM97 Q5BJF2 1/20 0.43
EBP Q15125 1/20 0.43
HTR2A P28223 1/20 0.43
HTR2C P28335 1/20 0.43
HTR2B P41595 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL432639 0.98 GAA (0.58) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL432356 0.94 GAA (0.53) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL433540 0.89 GAA (0.52) GAATSHRAGTR1HTR2AHTR2C
SCHEMBL3795015 0.85 CHRNB2 (0.55) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL126782 0.83 PTGDR2 (0.50) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL3793544 0.83 CHRNB2 (0.57) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL3786167 0.82 SLC6A2 (0.50) GAATSHRAGTR1CELSIGMAR1
SCHEMBL15566598 0.81 PTGDR2 (0.49) GAATSHRAGTR1PTGDR2PTGDR
SCHEMBL24736536 0.80 OPRL1 (0.48) PTGDR2CELSIGMAR1TMEM97EBP
SCHEMBL8331330 0.80 SLC6A2 (0.49) GAATSHRAGTR1CELSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104945309-A Novel nitroso compounds as nitroxyl donors and methods of use thereof CARDIOXYL PHARMACEUTICALS INC 2015-09-30 CN disclosed
CN-102076342-B Novel nitroso compounds as nitroxyl donors and methods of use thereof CARDIOXYL PHARMACEUTICALS INC 2015-06-10 CN disclosed
EP-2595984-A1 MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
EP-2595985-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES Syngenta Participations AG (CH) 2013-05-29 EP disclosed
WO-2012010567-A1 ISOXAZOLE, ISOTHIAZOLE, FURANE AND THIOPHENE COMPOUNDS AS MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
WO-2012010568-A1 MICROBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2012-01-26 WO disclosed
CN-102076342-A Novel nitroso compounds as nitroxyl donors and methods of use thereof CARDIOXYL PHARMACEUTICALS INC 2011-05-25 CN disclosed
US-4921935-A Preparation of polyarylene sulphides with ketone or pinacone BAYER AKTIENGESELLSCHAFT (DE) 1990-05-01 US disclosed