SCHEMBL4347126

SCHEMBL4347126

Cc1nc2ccc(C(=O)N3CC4(C)CN(C(=O)c5ccc6nc(C)c(C)nc6c5)CC(C)(C3)C4)cc2nc1C

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.53
MAPT P10636 4/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 8/20 0.43
KDM4E B2RXH2 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
KLK7 P49862 1/20 0.41
RAB9A P51151 1/20 0.41
CACNA1B Q00975 1/20 0.41
APBA1 Q02410 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
TP53 P04637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347243 0.85 MAPT (0.42) TDP1MAPTALDH1A1HPGDKDM4E
SCHEMBL4350146 0.85 TDP1 (0.51) TDP1MAPTALDH1A1HPGDKDM4E
SCHEMBL4346476 0.82 HPGD (0.61) TDP1MAPTALDH1A1HPGDRAB9A
SCHEMBL4356080 0.81 HPGD (0.41) MAPTALDH1A1HPGD
SCHEMBL4354045 0.78 KMT2A (0.44) TDP1MAPTALDH1A1HPGDKMT2A
SCHEMBL4351695 0.77 KDM4E (0.49) MAPTALDH1A1HPGDKDM4E
SCHEMBL16003043 0.72 HPGD (0.54) TDP1MAPTALDH1A1HPGDKDM4E
SCHEMBL4349007 0.71 KMT2A (0.41) TDP1MAPTALDH1A1HPGDKDM4E
SCHEMBL4342175 0.70 HPGD (0.62) ALDH1A1HPGDGAAKMT2ATP53
SCHEMBL4347843 0.70 HPGD (0.61) MAPTALDH1A1HPGDKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP claimed
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP disclosed