SCHEMBL4347601

SCHEMBL4347601

O=C(O)c1cc(NCc2cc([N+](=O)[O-])ccc2Sc2ccc(Cl)cc2)ccc1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
MAPT P10636 3/20 0.47
NOX4 Q9NPH5 2/20 0.47
ALDH1A1 P00352 2/20 0.47
EGFR P00533 2/20 0.47
TDP1 Q9NUW8 2/20 0.47
RGS12 O14924 1/20 0.47
LCK P06239 1/20 0.47
CAMKK2 Q96RR4 1/20 0.47
LDHA P00338 1/20 0.46
LDHB P07195 1/20 0.46
HAO1 Q9UJM8 1/20 0.46
POLB P06746 1/20 0.43
BCL2L1 Q07817 1/20 0.43
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
PLA2G1B P04054 1/20 0.43
ATG4B Q9Y4P1 1/20 0.43
APP P05067 1/20 0.42
IDO1 P14902 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6225219 0.95 NPC1 (0.46) NPC1MAPTNOX4ALDH1A1EGFR
SCHEMBL4350329 0.90 PTGES (0.48) NPC1MAPTNOX4ALDH1A1EGFR
SCHEMBL4345719 0.88 NPC1 (0.48) NPC1MAPTALDH1A1EGFRPOLB
SCHEMBL4351725 0.87 EGFR (0.53) NPC1MAPTALDH1A1EGFRTDP1
SCHEMBL6225218 0.87 NPC1 (0.41) NPC1MAPTNOX4ALDH1A1EGFR
SCHEMBL4351067 0.86 MAPT (0.47) NPC1MAPTALDH1A1EGFRPOLB
SCHEMBL4345711 0.86 NPC1 (0.49) NPC1MAPTALDH1A1EGFRPOLB
SCHEMBL4341720 0.85 NOX4 (0.58) MAPTNOX4ALDH1A1EGFRTDP1
SCHEMBL4345406 0.83 NOX4 (0.62) MAPTNOX4ALDH1A1EGFRTDP1
SCHEMBL27749183 0.82 EGFR (0.67) MAPTNOX4ALDH1A1EGFRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed