SCHEMBL4349130

SCHEMBL4349130

O=C(NCc1ccccc1)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.61
NPC1 O15118 4/20 0.61
POLB P06746 1/20 0.61
MAOB P27338 1/20 0.61
NAMPT P43490 1/20 0.55
HTT P42858 1/20 0.54
MEN1 O00255 1/20 0.54
TP53 P04637 1/20 0.54
HPGD P15428 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
MAPT P10636 1/20 0.54
ROCK2 O75116 2/20 0.52
ROCK1 Q13464 2/20 0.52
CA12 O43570 1/20 0.52
CA1 P00915 1/20 0.52
CA2 P00918 1/20 0.52
CA9 Q16790 1/20 0.52
GSK3B P49841 1/20 0.52
RORC P51449 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20804368 0.85 NPC1 (0.65) RAB9ANPC1POLBMAOBHTT
SCHEMBL4347762 0.85 NPC1 (0.59) RAB9ANPC1MEN1KMT2ASMN1; SMN2
SCHEMBL4357696 0.85 NAMPT (0.59) RAB9ANPC1POLBMAOBNAMPT
SCHEMBL4348348 0.83 MTOR (0.69) RAB9ANPC1POLBMAOBNAMPT
SCHEMBL4345336 0.82 MAOB (0.66) RAB9ANPC1POLBMAOBMEN1
SCHEMBL4350061 0.82 MTOR (0.55) RAB9ANPC1POLBMAOBHTT
SCHEMBL4347380 0.82 CA1 (0.56) RAB9ANPC1POLBMAOBNAMPT
SCHEMBL4350316 0.81 POLB (0.54) RAB9ANPC1POLBMAOBMEN1
SCHEMBL4350139 0.80 SMN1; SMN2 (0.63) RAB9ANPC1MAOBHTTMEN1
SCHEMBL4342163 0.80 RAB9A (0.61) RAB9ANPC1NAMPTHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed