SCHEMBL4348348

SCHEMBL4348348

O=C(NCc1ccc(C(F)(F)F)cc1)Nc1cc(F)c(O)c(F)c1

nearest known ligand 0.69

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MTOR P42345 4/20 0.69
NAMPT P43490 3/20 0.61
PRMT3 O60678 1/20 0.55
TRPV1 Q8NER1 2/20 0.53
NPC1 O15118 1/20 0.49
POLB P06746 1/20 0.49
MAOB P27338 1/20 0.49
RAB9A P51151 1/20 0.49
CNR1 P21554 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
MCHR1 Q99705 1/20 0.47
EPHX2 P34913 1/20 0.47
RORC P51449 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347646 0.87 MTOR (0.70) MTORNAMPTPRMT3TRPV1POLB
SCHEMBL4353993 0.85 MTOR (0.67) MTORNAMPTPRMT3TRPV1POLB
SCHEMBL4350068 0.85 MTOR (0.67) MTORNAMPTPRMT3TRPV1CNR1
SCHEMBL4341860 0.84 MEN1 (0.63) MTORMAOBMEN1KMT2A
SCHEMBL4347640 0.83 MTOR (0.57) MTORNAMPTPRMT3TRPV1NPC1
SCHEMBL4349130 0.83 RAB9A (0.61) NAMPTNPC1POLBMAOBRAB9A
SCHEMBL4345745 0.83 EPHX2 (0.71) MTORTRPV1RAB9AMEN1KMT2A
SCHEMBL4341854 0.81 MTOR (0.55) MTORNAMPTPRMT3TRPV1MEN1
SCHEMBL28808075 0.80 MTOR (0.76) MTORNAMPTPRMT3NPC1POLB
SCHEMBL26625460 0.80 MTOR (0.71) MTORNAMPTPRMT3TRPV1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed