SCHEMBL4347380

SCHEMBL4347380

O=C(NCc1ccccc1)Nc1cc(Br)c(O)c(Br)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.56
CA2 P00918 3/20 0.56
CA12 O43570 2/20 0.56
CA9 Q16790 2/20 0.56
NPC1 O15118 4/20 0.54
RAB9A P51151 4/20 0.54
POLB P06746 1/20 0.54
MAOB P27338 1/20 0.54
HTT P42858 1/20 0.54
MEN1 O00255 1/20 0.54
TP53 P04637 1/20 0.54
HPGD P15428 1/20 0.54
KMT2A Q03164 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
MAPT P10636 2/20 0.54
ROCK2 O75116 2/20 0.52
ROCK1 Q13464 2/20 0.52
GSK3B P49841 1/20 0.52
CFD P00746 1/20 0.50
IMPDH2 P12268 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20804368 0.85 NPC1 (0.65) CA1CA2CA12CA9NPC1
SCHEMBL4351660 0.85 NPC1 (0.59) CA1CA2CA12CA9NPC1
SCHEMBL4350068 0.82 MTOR (0.67) CA1CA2CA9MEN1KMT2A
SCHEMBL4345433 0.82 MAOB (0.66) CA9NPC1RAB9APOLBMAOB
SCHEMBL4349130 0.82 RAB9A (0.61) CA1CA2CA12CA9NPC1
SCHEMBL4350061 0.82 MTOR (0.55) CA1CA2CA12CA9NPC1
SCHEMBL4350351 0.80 SMN1; SMN2 (0.63) CA1CA2CA12CA9NPC1
SCHEMBL2831462 0.80 NPC1 (0.77) CA1CA2CA12CA9NPC1
SCHEMBL27942206 0.80 KMT2A (0.69) CA1CA2CA12CA9NPC1
SCHEMBL8177075 0.79 EGFR (0.65) NPC1RAB9APOLBMAOBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed