SCHEMBL4349923

SCHEMBL4349923

CN(C)CCN(C)C(=O)c1ccc(-c2ccc3c(c2)COC(C2CCN(C(=O)OC(C)(C)C)CC2)O3)cn1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 17/20 0.44
PTPN2 P17706 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN6 P29350 1/20 0.37
USP30 Q70CQ3 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4356487 0.89 ROCK2 (0.36) GPR119
SCHEMBL13586038 0.87 GPR119 (0.54) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL4352054 0.87 GPR119 (0.46) GPR119
SCHEMBL4355344 0.84 GPR119 (0.43) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL4521195 0.84 GPR119 (0.42) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL13586066 0.81 GPR119 (0.46) GPR119PTPN2PTPN1PTPN6
SCHEMBL4360506 0.81 GPR119 (0.47) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL4358492 0.80 GPR119 (0.53) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL4358178 0.80 GPR119 (0.51) GPR119PTPN2PTPN1PTPN6USP30
SCHEMBL4536702 0.78 GPR119 (0.49) GPR119PTPN2PTPN1PTPN6USP30

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO claimed
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO disclosed