SCHEMBL4351227

SCHEMBL4351227

CC(=O)C1Oc2ccc(C(=O)N3CC4(C)CN(C(=O)c5ccc6c(c5Cl)OC(C(C)=O)O6)CC(C)(C3)C4=O)c(Cl)c2O1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
ALDH1A1 P00352 3/20 0.33
MAPT P10636 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4345839 0.87 AVPR1A (0.33) GAAALDH1A1
SCHEMBL4346468 0.76 GAA (0.41) GAAALDH1A1TSHRKMT2A
SCHEMBL4341694 0.64 HPGD (0.42) GAAALDH1A1TSHRKMT2A
SCHEMBL4347434 0.63 GAA (0.48) GAAALDH1A1MAPTTSHRKMT2A
SCHEMBL4351639 0.60 HPGD (0.59) GAAALDH1A1MAPTTSHR
SCHEMBL4354898 0.59 GAA (0.40) GAAALDH1A1
SCHEMBL1856622 0.57 THRB (0.39) ALDH1A1
SCHEMBL3399484 0.56 POLB (0.45) GAAALDH1A1MAPTKMT2ANPC1
SCHEMBL4352206 0.56 GAA (0.39) GAAALDH1A1MAPTTSHRKMT2A
SCHEMBL31085036 0.55 ALDH1A1 (0.39) ALDH1A1TSHRKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP claimed
EP-2088149-A1 PHARMACOLOGICALLY ACTIVE N,N'-SUBSTITUTED 3,7-DIAZABICYCLO Ý3.3.1¨NONANES, PHARMACEUTICAL COMPOSITIONS BASED THEREON AND A METHOD FOR THE USE THEREOF Institute of Physiologically active compunds of the Russian Academy of Sciences (IPAC RAN) (RU) 2009-08-12 EP disclosed