SCHEMBL4351660

SCHEMBL4351660

O=C(NCCc1ccccc1)Nc1cc(Br)c(O)c(Br)c1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.59
RAB9A P51151 3/20 0.59
CNR1 P21554 3/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
HDAC1 Q13547 2/20 0.59
HDAC2 Q92769 2/20 0.59
MEN1 O00255 1/20 0.59
MAPT P10636 1/20 0.59
KMT2A Q03164 1/20 0.59
CA2 P00918 5/20 0.58
CA12 O43570 4/20 0.57
CA1 P00915 4/20 0.57
CA9 Q16790 4/20 0.57
EPHX1 P07099 3/20 0.56
KDM4E B2RXH2 1/20 0.56
ROCK2 O75116 1/20 0.54
ROCK1 Q13464 1/20 0.54
FPR2 P25090 1/20 0.52
PRMT3 O60678 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347380 0.85 CA1 (0.56) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL4347762 0.83 NPC1 (0.59) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL4351106 0.83 CNR1 (0.68) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL4350009 0.83 RAB9A (0.68) NPC1RAB9ASMN1; SMN2MEN1MAPT
SCHEMBL4606056 0.81 EPHX1 (0.81) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL4897395 0.81 CNR1 (0.74) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL28408741 0.80 KMT2A (0.71) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL8131908 0.79 NPC1 (0.62) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL22588919 0.78 KMT2A (0.72) NPC1RAB9ACNR1SMN1; SMN2HDAC1
SCHEMBL4350351 0.78 SMN1; SMN2 (0.63) NPC1RAB9ASMN1; SMN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed