SCHEMBL4351759

SCHEMBL4351759

CN1CCCN(C2(CNC(=O)c3cn(-c4ncccn4)c4cccc(Cl)c34)CCCCC2)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 4/20 0.60
P2RX7 Q99572 4/20 0.52
HCN1 O60741 5/20 0.52
TP53 P04637 3/20 0.49
IL1B P01584 3/20 0.48
OPRM1 P35372 2/20 0.47
SIGMAR1 Q99720 2/20 0.47
SLC6A9 P48067 5/20 0.46
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4357339 0.97 HCN4 (0.63) HCN4P2RX7HCN1TP53IL1B
SCHEMBL3688404 0.97 HCN4 (0.63) HCN4P2RX7HCN1TP53IL1B
SCHEMBL13706846 0.89 HCN4 (0.59) HCN4P2RX7HCN1TP53IL1B
SCHEMBL4537785 0.89 HCN4 (0.52) HCN4P2RX7HCN1IL1BSLC6A9
SCHEMBL4537218 0.89 HCN4 (0.54) HCN4P2RX7HCN1IL1BSLC6A9
SCHEMBL4530146 0.89 HCN4 (0.54) HCN4P2RX7HCN1IL1BSLC6A9
SCHEMBL13706814 0.89 HCN4 (0.51) HCN4P2RX7HCN1TP53IL1B
SCHEMBL4350608 0.89 HCN4 (0.55) HCN4P2RX7HCN1IL1BSLC6A9
SCHEMBL4361081 0.89 HCN4 (0.55) HCN4P2RX7HCN1IL1BSLC6A9
SCHEMBL4355954 0.88 HCN1 (0.62) HCN4P2RX7HCN1TP53OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed