SCHEMBL4355954

SCHEMBL4355954

Cc1cccc2c1c(C(=O)NCC1(N3CCN(C)CC3)CCCCC1)cn2-c1ncccn1

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCN1 O60741 6/20 0.62
HCN4 Q9Y3Q4 6/20 0.54
THRB P10828 3/20 0.54
TP53 P04637 4/20 0.52
OPRM1 P35372 2/20 0.50
SIGMAR1 Q99720 2/20 0.50
ALDH1A1 P00352 1/20 0.46
TSHR P16473 1/20 0.46
LMNA P02545 4/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
P2RX7 Q99572 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535037 0.91 HCN4 (0.55) HCN1HCN4THRBTP53ALDH1A1
SCHEMBL4364182 0.91 HCN4 (0.56) HCN1HCN4THRBTP53ALDH1A1
SCHEMBL3688404 0.90 HCN4 (0.63) HCN1HCN4THRBTP53OPRM1
SCHEMBL4357339 0.90 HCN4 (0.63) HCN1HCN4THRBTP53OPRM1
SCHEMBL4355970 0.90 HCN1 (0.54) HCN1HCN4THRBTP53OPRM1
SCHEMBL4351759 0.88 HCN4 (0.60) HCN1HCN4THRBTP53OPRM1
SCHEMBL13706853 0.88 HCN1 (0.60) HCN1HCN4THRBTP53OPRM1
SCHEMBL13706779 0.85 HCN1 (0.57) HCN1HCN4THRBTP53OPRM1
SCHEMBL13706601 0.85 HCN1 (0.44) HCN1HCN4THRBTP53ALDH1A1
SCHEMBL4540375 0.85 HCN1 (0.44) HCN1HCN4THRBTP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed