SCHEMBL4353663

SCHEMBL4353663

O=C(Nc1ccc(Cl)cc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.60
KMT2A Q03164 6/20 0.60
HTT P42858 4/20 0.60
LMNA P02545 3/20 0.60
NPC1 O15118 3/20 0.60
EPHX2 P34913 2/20 0.60
EPHX1 P07099 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
CHRM1 P11229 1/20 0.60
SLC6A2 P23975 1/20 0.60
PDE4A P27815 1/20 0.60
ADRA1A P35348 1/20 0.60
OPRM1 P35372 1/20 0.60
PDE3A Q14432 1/20 0.60
NLRP3 Q96P20 1/20 0.60
SLC2A1 P11166 1/20 0.57
RAB9A P51151 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
MAPT P10636 4/20 0.55
CNR1 P21554 5/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4347321 0.89 P2RY1 (0.61) MEN1KMT2AHTTLMNANPC1
SCHEMBL4351601 0.85 MAOA (0.59) MEN1KMT2AHTTLMNANPC1
SCHEMBL4348841 0.85 MEN1 (0.57) MEN1KMT2AHTTLMNANPC1
SCHEMBL14758363 0.85 MEN1 (0.72) MEN1KMT2AHTTLMNANPC1
SCHEMBL4348076 0.83 MEN1 (0.62) MEN1KMT2AHTTLMNANPC1
SCHEMBL4345497 0.83 MEN1 (0.74) MEN1KMT2AHTTLMNANPC1
SCHEMBL4548132 0.82 IDH1 (0.64) MEN1KMT2AHTTLMNANPC1
SCHEMBL11048619 0.80 MEN1 (0.76) MEN1KMT2AHTTLMNANPC1
SCHEMBL4741253 0.80 MEN1 (0.76) MEN1KMT2AHTTLMNANPC1
SCHEMBL4357636 0.80 MAPT (0.61) MEN1KMT2AHTTLMNAEPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed