SCHEMBL4351601

SCHEMBL4351601

O=C(Nc1ccccc1)Nc1ccc(O)c(F)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.59
MAOB P27338 2/20 0.59
SMN1; SMN2 Q16637 5/20 0.59
TP53 P04637 2/20 0.59
EPHX1 P07099 1/20 0.59
TSHR P16473 1/20 0.59
EPHX2 P34913 1/20 0.59
CDK9 P50750 1/20 0.59
CLK4 Q9HAZ1 1/20 0.59
KMT2A Q03164 8/20 0.57
MEN1 O00255 6/20 0.57
MAPT P10636 5/20 0.57
HTT P42858 5/20 0.57
LMNA P02545 4/20 0.57
RAB9A P51151 7/20 0.57
NPC1 O15118 6/20 0.57
CASP3 P42574 1/20 0.56
SENP7 Q9BQF6 1/20 0.56
POLB P06746 1/20 0.54
ALDH1A1 P00352 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6229951 0.90 CA12 (0.60) SMN1; SMN2TP53TSHRKMT2AMEN1
SCHEMBL4352985 0.88 CA12 (0.58) SMN1; SMN2EPHX1KMT2AMEN1MAPT
SCHEMBL4353663 0.85 MEN1 (0.60) SMN1; SMN2EPHX1EPHX2KMT2AMEN1
SCHEMBL13772128 0.84 ALOX15 (0.71) MAOAMAOBSMN1; SMN2TP53EPHX1
SCHEMBL4345620 0.83 KMT2A (0.59) MAOAMAOBSMN1; SMN2TP53KMT2A
SCHEMBL4350139 0.82 SMN1; SMN2 (0.63) MAOAMAOBSMN1; SMN2TP53EPHX1
SCHEMBL1962890 0.82 NPC1 (0.47) SMN1; SMN2TP53EPHX2KMT2AMEN1
SCHEMBL4357696 0.82 NAMPT (0.59) MAOBSMN1; SMN2TP53KMT2AMEN1
SCHEMBL4346828 0.82 DDX3X (0.66) SMN1; SMN2KMT2AMEN1MAPTHTT
SCHEMBL4122903 0.81 NPC1 (0.71) SMN1; SMN2TP53EPHX1TSHREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2022045365-A1 POLYPEPTIDE CONTAINING FIBRONECTIN TYPE III DOMAIN SCAFFOLD 国立大学法人東海国立大学機構 2022-03-03 WO disclosed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed