SCHEMBL4348453

SCHEMBL4348453

CC(O)c1cc(N(S)C(=O)Nc2ccc(C(F)(F)F)cc2)cc(Cl)c1O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.42
P2RX1 P51575 2/20 0.39
P2RX4 Q99571 2/20 0.39
P2RX7 Q99572 2/20 0.39
TMPRSS4 Q9NRS4 2/20 0.39
MTOR P42345 1/20 0.38
EPHX2 P34913 1/20 0.38
UTS2R Q9UKP6 2/20 0.37
CNR2 P34972 1/20 0.37
LMNA P02545 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TRPV1 Q8NER1 1/20 0.37
HTT P42858 1/20 0.37
KCNJ5 P48544 1/20 0.37
KCNJ3 P48549 1/20 0.37
BAZ1A Q9NRL2 1/20 0.36
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355433 0.88 TSHR (0.43) EPHX2LMNASMN1; SMN2HTT
SCHEMBL4359460 0.88 EPHX2 (0.46) P2RX1P2RX4P2RX7TMPRSS4MTOR
SCHEMBL4354101 0.85 SMN1; SMN2 (0.39) MTORLMNASMN1; SMN2HTT
SCHEMBL4354911 0.85 PDE2A (0.40) PDE2AMTOREPHX2
SCHEMBL4341759 0.83 P2RX1 (0.41) PDE2AP2RX1P2RX4P2RX7TMPRSS4
SCHEMBL4354080 0.82 ALDH1A1 (0.36) P2RX1P2RX4P2RX7TMPRSS4SMN1; SMN2
SCHEMBL4349857 0.81 POLB (0.41) SMN1; SMN2TRPV1HTT
SCHEMBL4346902 0.80 EPHX2 (0.54) PDE2AP2RX1P2RX4P2RX7TMPRSS4
SCHEMBL4341321 0.78 P2RX1 (0.50) P2RX1P2RX4P2RX7TMPRSS4MTOR
SCHEMBL4358931 0.78 EPHX2 (0.49) P2RX1P2RX4P2RX7TMPRSS4MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed