SCHEMBL4354080

SCHEMBL4354080

CC(O)c1cc(N(S)C(=O)Nc2cc(Cl)cc(Cl)c2)cc(Cl)c1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 2/20 0.34
P2RY1 P47900 1/20 0.33
STK39 Q9UEW8 2/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
PTGS1 P23219 1/20 0.33
TBXAS1 P24557 1/20 0.33
MAPK1 P28482 1/20 0.33
PTGS2 P35354 1/20 0.33
MAPK14 Q16539 1/20 0.33
GRM4 Q14833 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.32
P2RX1 P51575 1/20 0.32
P2RX4 Q99571 1/20 0.32
P2RX7 Q99572 1/20 0.32
TMPRSS4 Q9NRS4 1/20 0.32
ACLY P53396 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4355433 0.89 TSHR (0.43) ALDH1A1SMN1; SMN2GAASTK39MEN1
SCHEMBL4354101 0.87 SMN1; SMN2 (0.39) ALDH1A1SMN1; SMN2GAASTK39MEN1
SCHEMBL4342472 0.86 P2RY1 (0.41) ALDH1A1P2RY1STK39MEN1KMT2A
SCHEMBL4350861 0.82 ALDH1A1 (0.38) ALDH1A1SMN1; SMN2GAAP2RY1MEN1
SCHEMBL4351937 0.82 MAPK1 (0.33) ALDH1A1GAAMEN1KMT2AMAPK1
SCHEMBL4348453 0.82 PDE2A (0.42) SMN1; SMN2P2RX1P2RX4P2RX7TMPRSS4
SCHEMBL4348034 0.76 MEN1 (0.38) ALDH1A1P2RY1MEN1KMT2AGRM4
SCHEMBL4349857 0.76 POLB (0.41) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL4347618 0.75 PKM (0.39) ALDH1A1SMN1; SMN2GAAMEN1KMT2A
SCHEMBL4351425 0.75 EPHX2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed