SCHEMBL4354464

SCHEMBL4354464

CC(=O)c1cc(NCc2ccccc2Sc2cccc(Cl)c2)cc(Cl)c1O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.46
SLC6A4 P31645 1/20 0.46
SLC6A3 Q01959 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.43
SLC6A9 P48067 4/20 0.38
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KCNJ5 P48544 1/20 0.37
KCNJ3 P48549 1/20 0.37
TP53 P04637 1/20 0.36
CPT2 P23786 1/20 0.35
CPT1A P50416 1/20 0.35
CPT1B Q92523 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4343453 0.92 SMN1; SMN2 (0.43) SMN1; SMN2KDM4EMEN1MAPTCYP2C9
SCHEMBL4346923 0.90 SLC6A4 (0.43) SLC6A2SLC6A4SLC6A3SMN1; SMN2KDM4E
SCHEMBL4348911 0.89 MEN1 (0.39) SMN1; SMN2MEN1MAPTCYP2C9CYP2C19
SCHEMBL4354940 0.88 SLC6A4 (0.52) SLC6A2SLC6A4SLC6A3SMN1; SMN2SLC6A9
SCHEMBL4351627 0.87 MAPT (0.39) SLC6A2SLC6A4SLC6A3SMN1; SMN2MEN1
SCHEMBL4344018 0.86 DHODH (0.38) SMN1; SMN2KDM4EMEN1CYP3A4MAPT
SCHEMBL4351090 0.85 LMNA (0.41) SMN1; SMN2SLC6A9KDM4ECYP3A4MAPT
SCHEMBL4354650 0.84 SLC6A2 (0.47) SLC6A2SLC6A4SLC6A3SMN1; SMN2SLC6A9
SCHEMBL4347108 0.84 KMT2A (0.50) SMN1; SMN2KDM4EMEN1CYP3A4MAPT
SCHEMBL4357651 0.82 MAPT (0.43) SMN1; SMN2MEN1CYP3A4MAPTCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed