SCHEMBL4343453

SCHEMBL4343453

CC(=O)c1cc(NCc2ccccc2Sc2ccccc2)cc(Cl)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
NOX4 Q9NPH5 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP2D6 P10635 1/20 0.39
DHODH Q02127 1/20 0.38
EGFR P00533 1/20 0.37
RAB9A P51151 1/20 0.37
GFER P55789 1/20 0.37
ALDH1A1 P00352 2/20 0.36
HPGD P15428 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
G6PD P11413 1/20 0.36
PKM P14618 1/20 0.36
MAPK1 P28482 1/20 0.36
RECQL P46063 1/20 0.36
CCR6 P51684 1/20 0.36
MCL1 Q07820 1/20 0.36
HKDC1 Q2TB90 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346923 0.94 SLC6A4 (0.43) SMN1; SMN2NOX4CYP2C9CYP2C19CYP2D6
SCHEMBL4351627 0.93 MAPT (0.39) SMN1; SMN2NOX4CYP2C9CYP2C19CYP2D6
SCHEMBL4354464 0.92 SLC6A2 (0.46) SMN1; SMN2NOX4CYP2C9CYP2C19DHODH
SCHEMBL4351090 0.91 LMNA (0.41) SMN1; SMN2NOX4CYP2C9CYP2C19CYP2D6
SCHEMBL4348911 0.90 MEN1 (0.39) SMN1; SMN2NOX4CYP2C9CYP2C19CYP2D6
SCHEMBL4344018 0.90 DHODH (0.38) SMN1; SMN2NOX4CYP2C9CYP2C19DHODH
SCHEMBL4347108 0.90 KMT2A (0.50) SMN1; SMN2NOX4CYP2C9CYP2C19EGFR
SCHEMBL4357651 0.88 MAPT (0.43) SMN1; SMN2CYP2C9CYP2C19CYP2D6ALDH1A1
SCHEMBL4351063 0.87 SMN1; SMN2 (0.43) SMN1; SMN2CYP2C9CYP2C19CYP2D6RAB9A
SCHEMBL4347491 0.83 CTSD (0.40) SMN1; SMN2RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed