SCHEMBL4354589

SCHEMBL4354589

O=C(Nc1ccc(Oc2ccccc2)cc1)Nc1ccc(O)c(Cl)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.61
KMT2A Q03164 4/20 0.61
MAPT P10636 3/20 0.61
LMNA P02545 3/20 0.61
NPSR1 Q6W5P4 1/20 0.61
CA12 O43570 5/20 0.58
CA1 P00915 5/20 0.58
CA2 P00918 5/20 0.58
CA9 Q16790 5/20 0.58
STK39 Q9UEW8 1/20 0.55
P2RY1 P47900 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
NPC1 O15118 2/20 0.55
HTT P42858 1/20 0.55
PNLIP P16233 3/20 0.54
RNF4 P78317 1/20 0.52
POLB P06746 1/20 0.52
GAA P10253 1/20 0.52
RAB9A P51151 1/20 0.52
HPGD P15428 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6252145 0.99 CA12 (0.60) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL4358566 0.88 MEN1 (0.69) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL4350770 0.87 MEN1 (0.67) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL4352985 0.83 CA12 (0.58) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL30053559 0.83 CA12 (0.73) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL4358450 0.82 CA12 (0.68) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL6229951 0.82 CA12 (0.60) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL13556607 0.82 NPC1 (0.62) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL21295379 0.81 PNLIP (0.66) MEN1KMT2AMAPTLMNANPSR1
SCHEMBL21295380 0.81 CA12 (0.71) MEN1KMT2AMAPTLMNANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed