SCHEMBL4358566

SCHEMBL4358566

O=C(Nc1ccccc1)Nc1ccc(O)c(Cl)c1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 9/20 0.69
KMT2A Q03164 9/20 0.69
MAPT P10636 7/20 0.69
NPC1 O15118 6/20 0.69
LMNA P02545 5/20 0.69
HTT P42858 4/20 0.69
SMN1; SMN2 Q16637 3/20 0.69
RAB9A P51151 5/20 0.62
GAA P10253 3/20 0.60
POLB P06746 3/20 0.60
EPHX1 P07099 3/20 0.59
EPHX2 P34913 3/20 0.59
MAOA P21397 1/20 0.59
MAOB P27338 1/20 0.59
NPSR1 Q6W5P4 2/20 0.59
TP53 P04637 1/20 0.59
TSHR P16473 1/20 0.59
CDK9 P50750 1/20 0.59
CLK4 Q9HAZ1 1/20 0.59
CNR1 P21554 3/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6252145 0.90 CA12 (0.60) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4354589 0.88 MEN1 (0.61) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4345497 0.88 MEN1 (0.74) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL7980937 0.86 EPHX1 (0.81) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL13772128 0.84 ALOX15 (0.71) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4343605 0.83 KMT2A (0.59) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL12499571 0.83 P2RY1 (0.75) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4342381 0.82 KMT2A (0.68) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4683057 0.82 MAPT (0.55) MEN1KMT2AMAPTNPC1LMNA
SCHEMBL4360021 0.82 DDX3X (0.66) MEN1KMT2AMAPTNPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2022045365-A1 POLYPEPTIDE CONTAINING FIBRONECTIN TYPE III DOMAIN SCAFFOLD 国立大学法人東海国立大学機構 2022-03-03 WO disclosed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed