SCHEMBL4354905

SCHEMBL4354905

CC(O)c1cc(NC(=S)NCc2ccc(C(F)(F)F)cc2)cc(Cl)c1O

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 10/20 0.51
MEN1 O00255 9/20 0.51
KMT2A Q03164 9/20 0.51
ALDH1A1 P00352 7/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
HTT P42858 3/20 0.51
GAA P10253 3/20 0.51
NPSR1 Q6W5P4 2/20 0.51
MYC P01106 1/20 0.50
MAX P61244 1/20 0.50
LMNA P02545 6/20 0.47
HPGD P15428 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
MAPK1 P28482 1/20 0.46
PDE2A O00408 1/20 0.42
ALOX12 P18054 2/20 0.41
BLM P54132 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4357497 0.88 MEN1 (0.61) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4347012 0.87 MTOR (0.56)
SCHEMBL4348451 0.87 PDE2A (0.48) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4342192 0.85 MAPT (0.53) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL6225190 0.84 MAPT (0.48) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4345508 0.83 KMT2A (0.48) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4357659 0.78 MAPT (0.62) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4346902 0.78 EPHX2 (0.54) MAPTMEN1KMT2AHTTPDE2A
SCHEMBL4341860 0.77 MEN1 (0.63) MAPTMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL4345459 0.76 MEN1 (0.46) MAPTMEN1KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed