SCHEMBL4342192

SCHEMBL4342192

CC(O)c1cc(NC(=S)NCc2ccccc2)cc(Cl)c1O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HPGD P15428 3/20 0.53
MAOB P27338 3/20 0.53
LMNA P02545 2/20 0.53
PLA2G1B P04054 1/20 0.53
ATG4B Q9Y4P1 1/20 0.53
SMN1; SMN2 Q16637 3/20 0.53
ALOX12 P18054 2/20 0.53
ALDH1A1 P00352 1/20 0.53
HTT P42858 1/20 0.53
MAOA P21397 1/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
RAB9A P51151 2/20 0.49
POLB P06746 2/20 0.49
MYC P01106 1/20 0.49
MAX P61244 1/20 0.49
NPC1 O15118 1/20 0.48
CYP19A1 P11511 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4350105 0.88 MAPT (0.55) MAPTHPGDMAOBLMNAPLA2G1B
SCHEMBL6226369 0.87 LMNA (0.48) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL4355796 0.86 MAPT (0.66) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL4354905 0.85 MAPT (0.51) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL4345459 0.85 MEN1 (0.46) MAPTNPSR1HPGDLMNASMN1; SMN2
SCHEMBL4354098 0.85 ALDH1A1 (0.47) MAPTHPGDMAOBLMNASMN1; SMN2
SCHEMBL4351070 0.81 SMN1; SMN2 (0.56) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL26485863 0.79 MAPT (0.64) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL4351932 0.79 KDM4E (0.41) MAPTNPSR1HPGDMAOBLMNA
SCHEMBL27782816 0.78 SMN1; SMN2 (0.52) MAPTNPSR1HPGDLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed