SCHEMBL4345459

SCHEMBL4345459

Cc1ccccc1CNC(=S)Nc1cc(Cl)c(O)c(C(C)O)c1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
LMNA P02545 5/20 0.46
ALOX12 P18054 4/20 0.46
MAPT P10636 4/20 0.46
ALDH1A1 P00352 4/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
PPARG P37231 2/20 0.44
NCOA3 Q9Y6Q9 1/20 0.44
HPGD P15428 1/20 0.43
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PKM P14618 1/20 0.41
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
DHODH Q02127 1/20 0.40
QPCT Q16769 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6226369 0.90 LMNA (0.48) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4348819 0.88 MEN1 (0.54) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4354116 0.87 NPC1 (0.58) MEN1KMT2AMAPTALDH1A1PPARG
SCHEMBL4342192 0.85 MAPT (0.53) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4347975 0.82 ALOX12 (0.51) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4354098 0.80 ALDH1A1 (0.47) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL6672908 0.79 EPHX2 (0.52) ALDH1A1HTTNPC1RAB9A
SCHEMBL4357807 0.79 MAPT (0.54) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4350105 0.79 MAPT (0.55) MEN1KMT2ALMNAALOX12MAPT
SCHEMBL4351932 0.76 KDM4E (0.41) MEN1KMT2ALMNAALOX12MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed