SCHEMBL4347012

SCHEMBL4347012

CC(O)c1cc(NC(=O)NCc2ccc(C(F)(F)F)cc2)cc(Cl)c1O

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MTOR P42345 3/20 0.56
NAMPT P43490 2/20 0.50
PRMT3 O60678 1/20 0.46
RORC P51449 6/20 0.46
CNR1 P21554 1/20 0.45
TRPV1 Q8NER1 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA7 P43166 1/20 0.44
CA9 Q16790 1/20 0.44
MCHR1 Q99705 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRL1 P41146 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4353993 0.88 MTOR (0.67) MTORNAMPTPRMT3RORCCNR1
SCHEMBL4354905 0.87 MAPT (0.51)
SCHEMBL4346902 0.87 EPHX2 (0.54) MTORCA1CA2CA9
SCHEMBL4348962 0.83 MTOR (0.50) MTORNAMPTPRMT3CNR1TRPV1
SCHEMBL4348431 0.78 MTOR (0.68) MTORNAMPTPRMT3RORCCNR1
SCHEMBL4354911 0.78 PDE2A (0.40) MTOROPRM1OPRL1
SCHEMBL4348451 0.78 PDE2A (0.48) CA1CA2CA9
SCHEMBL4348348 0.77 MTOR (0.69) MTORNAMPTPRMT3RORCCNR1
SCHEMBL6229028 0.77 MTOR (0.56) MTORNAMPTPRMT3RORCCNR1
SCHEMBL4354116 0.76 NPC1 (0.58) NAMPTRORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100546977-C Suppress the new compound and the application thereof of rotamase JERINI AG (DE) 2009-10-07 CN claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
CN-1701061-A Novel compounds for inhibiting rotamase enzymes and uses thereof JERINI AG (DE) 2005-11-23 CN claimed
WO-2004030664-A2 NEW COMPOUNDS FOR THE INHIBITION OF UNDESIRED CELL PROLIFERATION AND USE THEREOF JERINI AG (DE) 2004-04-15 WO claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed