SCHEMBL4355356

SCHEMBL4355356

O=C(Nc1ccccc1)N(S)c1cc(Br)c(O)c(Br)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSPD1 P10809 1/20 0.49
HSPE1 P61604 1/20 0.49
CDK9 P50750 2/20 0.47
CLK4 Q9HAZ1 2/20 0.47
CHEK1 O14757 1/20 0.47
AURKA O14965 1/20 0.47
DAPK3 O43293 1/20 0.47
JAK2 O60674 1/20 0.47
PRKD3 O94806 1/20 0.47
MAP4K4 O95819 1/20 0.47
PAK4 O96013 1/20 0.47
ABL1 P00519 1/20 0.47
NTRK1 P04629 1/20 0.47
LCK P06239 1/20 0.47
CSF1R P07333 1/20 0.47
RET P07949 1/20 0.47
IGF1R P08069 1/20 0.47
MET P08581 1/20 0.47
PDGFRB P09619 1/20 0.47
PIM1 P11309 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346608 0.85 TSHR (0.47) LCKEGFRERBB2MEN1KMT2A
SCHEMBL4341297 0.83 KMT2A (0.43) CDK9CLK4EGFRERBB2MEN1
SCHEMBL4353865 0.82 EPHX2 (0.46) MEN1KMT2AMAPTNPC1SMN1; SMN2
SCHEMBL4351896 0.82 MAPT (0.48) CDK9CLK4EGFRERBB2MEN1
SCHEMBL4349869 0.81 MEN1 (0.39) HSPD1HSPE1MEN1KMT2AALDH1A1
SCHEMBL5353973 0.80 MEN1 (0.56) CDK9CLK4MEN1KMT2AALDH1A1
SCHEMBL4349028 0.77 SMN1; SMN2 (0.50) MEN1KMT2AALDH1A1MAPTMAPK1
SCHEMBL4350012 0.76 HDAC2 (0.47) ALDH1A1NPC1RAB9AEPHX1
SCHEMBL4348538 0.74 NPC1 (0.47) HSPD1HSPE1PTK2EGFRERBB2
SCHEMBL9243026 0.74 CASP3 (0.56) MEN1KMT2AALDH1A1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed