SCHEMBL4349869

SCHEMBL4349869

O=C(Nc1cc(Cl)cc(Cl)c1)N(S)c1cc(Br)c(O)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 3/20 0.39
NPSR1 Q6W5P4 3/20 0.39
POLB P06746 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GLA P06280 1/20 0.39
CRHBP P24387 1/20 0.39
RECQL P46063 1/20 0.39
CRHR2 Q13324 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
HSPD1 P10809 1/20 0.37
HSPE1 P61604 1/20 0.37
RAB9A P51151 1/20 0.37
P2RX1 P51575 1/20 0.37
P2RX4 Q99571 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4346608 0.87 TSHR (0.47) MEN1MAPTKMT2AALDH1A1GAA
SCHEMBL4342472 0.85 P2RY1 (0.41) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL4348034 0.84 MEN1 (0.38) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL4355356 0.81 HSPD1 (0.49) MEN1MAPTKMT2ANPSR1ALDH1A1
SCHEMBL4350724 0.76 MEN1 (0.58) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL11194705 0.76 P2RX1 (0.42) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL4341619 0.75 P2RX1 (0.46) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL4353865 0.75 EPHX2 (0.46) MEN1MAPTKMT2ANPSR1RAB9A
SCHEMBL4357681 0.75 KMT2A (0.36) MEN1MAPTKMT2ANPSR1POLB
SCHEMBL4354080 0.75 ALDH1A1 (0.36) MEN1MAPTKMT2ANPSR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed