SCHEMBL4355874

SCHEMBL4355874

CC(C)(C)CC(C)(C)NC(=O)N(S)c1cc(Br)c(O)c(Br)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.37
HIF1A Q16665 3/20 0.35
TSHR P16473 2/20 0.35
HSD17B10 Q99714 2/20 0.35
CYP2C9 P11712 2/20 0.35
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
ALOX12 P18054 1/20 0.34
CASP1 P29466 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTT P42858 3/20 0.33
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4351219 0.84 POLB (0.38) POLBALDH1A1HPGDHTTMAPT
SCHEMBL4345693 0.83 POLB (0.37) POLBALDH1A1HPGDHTTMAPT
SCHEMBL4350397 0.76 POLB (0.34) POLBALDH1A1HPGDHTTMAPT
SCHEMBL4343914 0.75 POLB (0.32) POLB
SCHEMBL4342228 0.75 CA2 (0.42) POLBALDH1A1HPGDCYP3A4CASP1
SCHEMBL4351873 0.75 POLB (0.38) POLBHSD17B10ALDH1A1HPGDHTT
SCHEMBL4346754 0.72 POLB (0.50) POLBHIF1ATSHRHSD17B10CYP2C9
SCHEMBL4358520 0.72 AKR1C4 (0.36) POLBHIF1ATSHRHSD17B10ALDH1A1
SCHEMBL4345611 0.72 MAPT (0.42) POLBTSHRHSD17B10ALDH1A1HPGD
SCHEMBL4347757 0.72 PTGES (0.36) HIF1ATSHRHSD17B10CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed