SCHEMBL4347757

SCHEMBL4347757

CC(C)NC(=O)N(S)c1cc(Br)c(O)c(Br)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 2/20 0.36
FOLH1 Q04609 1/20 0.35
TTR P02766 1/20 0.35
TSHR P16473 3/20 0.32
CYP3A4 P08684 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
RECQL P46063 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HIF1A Q16665 2/20 0.32
HSD17B10 Q99714 2/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
ALOX12 P18054 1/20 0.32
CASP1 P29466 1/20 0.32
MAPK1 P28482 1/20 0.31
LMNA P02545 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4351134 0.82 ERN1 (0.36) PTGESALDH1A1HPGDLMNAALOX5
SCHEMBL4351937 0.74 MAPK1 (0.33) ALDH1A1MAPK1MAPT
SCHEMBL4351731 0.73 PTGES (0.36) PTGESALDH1A1MAPK1MAOAMAOB
SCHEMBL4350103 0.73 PKM (0.43) TSHRALDH1A1HSD17B10HPGDCYP2C9
SCHEMBL4355356 0.72 HSPD1 (0.49) TSHRALDH1A1HSD17B10ALOX15MAPK1
SCHEMBL4350363 0.72 TRPV1 (0.43) HPGD
SCHEMBL4355874 0.72 POLB (0.37) TTRTSHRCYP3A4TDP1RECQL
SCHEMBL4343483 0.71 ESR1 (0.39) PTGESFOLH1ALDH1A1HSD17B10LMNA
SCHEMBL4349869 0.71 MEN1 (0.39) TDP1RECQLALDH1A1KDM4EMAPT
SCHEMBL4357469 0.71 MAPK1 (0.38) TSHRALDH1A1HSD17B10MAPK1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP claimed
EP-2100876-A2 New compounds for the inhibition of rotamases and use thereof Jerini AG (DE) 2009-09-16 EP disclosed